SCHEMBL3873907

SCHEMBL3873907

Cc1nc([AsH2])c(C(N)=O)nc1-c1noc(C(C)(C)C)n1

nearest known ligand 0.34

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 3/20 0.34
CNR1 P21554 1/20 0.34
AOC3 Q16853 2/20 0.32
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
LMNA P02545 1/20 0.32
HPGD P15428 1/20 0.32
TSHR P16473 1/20 0.32
HSD17B10 Q99714 1/20 0.32
HDAC1 Q13547 1/20 0.31
HDAC8 Q9BY41 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31
DGAT1 O75907 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2678063 0.68 DPP4 (0.38) AOC3KDM4EALDH1A1LMNAHPGD
Hydrochloric Acid SCHEMBL23114008 0.67 DPP4 (0.37)
SCHEMBL3873906 0.65 CNR2 (0.39) CNR2CNR1AOC3HDAC6
Trifluoroacetic Acid SCHEMBL29279144 0.64 DPP4 (0.36)
SCHEMBL3467030 0.61 NPC1 (0.43) KDM4EALDH1A1LMNATSHRHSD17B10
SCHEMBL3873902 0.61 HDAC4 (0.41) CNR2HDAC1HDAC8HDAC6
Potassium Ion SCHEMBL20532715 0.60 DPP4 (0.37)
SCHEMBL15472482 0.60 IKBKB (0.40) KDM4EALDH1A1LMNAHSD17B10
SCHEMBL8965367 0.60 DPP4 (0.39) KDM4EALDH1A1LMNAHPGDTSHR
SCHEMBL19449365 0.60 DPP4 (0.39) KDM4EALDH1A1LMNAHPGDTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501514-A4 PROTEIN KINASE MODULATORS AND METHODS OF USE EXELIXIS INC (US) 2009-08-26 EP disclosed
EP-1501514-A2 PROTEIN KINASE MODULATORS AND METHODS OF USE Exelixis, Inc. (US) 2005-02-02 EP disclosed
WO-2003093297-A2 PROTEIN KINASE MODULATORS AND METHODS OF USE EXELIXIS, INC. (US) 2003-11-13 WO disclosed