SCHEMBL3873906

SCHEMBL3873906

CC(C)(C)c1nc(-c2cnc(C[AsH2])c(C(N)=O)n2)no1

nearest known ligand 0.39

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 17/20 0.39
HDAC4 P56524 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
CNR1 P21554 1/20 0.35
AOC3 Q16853 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3461135 0.72 PIK3CD (0.47) CNR2HDAC4HDAC6
SCHEMBL3873902 0.72 HDAC4 (0.41) CNR2HDAC4HDAC6
SCHEMBL3873907 0.65 CNR2 (0.34) CNR2HDAC6CNR1AOC3
SCHEMBL20043166 0.65 CNR2 (0.48) CNR2HDAC4HDAC6CNR1
SCHEMBL14349571 0.62 NPC1 (0.50) CNR2
SCHEMBL2678063 0.62 DPP4 (0.38) AOC3
SCHEMBL29625962 0.62 HDAC6 (0.60) HDAC4HDAC6
SCHEMBL16115983 0.61 CNR2 (0.65) CNR2CNR1
Hydrochloric Acid SCHEMBL23114008 0.60 DPP4 (0.37)
SCHEMBL16543467 0.59 RAB9A (0.61)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501514-A4 PROTEIN KINASE MODULATORS AND METHODS OF USE EXELIXIS INC (US) 2009-08-26 EP disclosed
EP-1501514-A2 PROTEIN KINASE MODULATORS AND METHODS OF USE Exelixis, Inc. (US) 2005-02-02 EP disclosed
WO-2003093297-A2 PROTEIN KINASE MODULATORS AND METHODS OF USE EXELIXIS, INC. (US) 2003-11-13 WO disclosed