SCHEMBL3876034

SCHEMBL3876034

CN(CCO)c1nc(-c2ccc(F)c(Cl)c2)cc(N2CCN(c3ncccc3C(F)(F)F)CC2)n1

nearest known ligand 0.44

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 5/20 0.44
HSD11B1 P28845 5/20 0.41
TRPA1 O75762 1/20 0.39
GALR2 O43603 1/20 0.39
GALR1 P47211 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13761373 0.91 TRPV1 (0.45) TRPV1HSD11B1GALR2GALR1
SCHEMBL3878651 0.90 HSD11B1 (0.43) TRPV1HSD11B1TRPA1GALR2GALR1
SCHEMBL3881354 0.89 TRPV1 (0.48) TRPV1HSD11B1GALR2GALR1
SCHEMBL3878894 0.89 HSD11B1 (0.42) TRPV1HSD11B1TRPA1
SCHEMBL13761395 0.89 HSD11B1 (0.43) TRPV1HSD11B1GALR2GALR1
SCHEMBL3889392 0.88 HSD11B1 (0.47) TRPV1HSD11B1GALR2GALR1
SCHEMBL3879463 0.87 HSD11B1 (0.42) TRPV1HSD11B1TRPA1GALR2GALR1
SCHEMBL3880107 0.87 HSD11B1 (0.43) HSD11B1GALR2GALR1
SCHEMBL3887131 0.87 TRPV1 (0.41) TRPV1HSD11B1TRPA1GALR2GALR1
SCHEMBL3878643 0.86 TRPA1 (0.43) TRPV1HSD11B1TRPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7566712-B2 Biaryl piperazinyl-pyridine analogues NEUROGEN CORPORATION (US) 2009-07-28 US disclosed
US-7566712-B2 Biaryl piperazinyl-pyridine analogues NEUROGEN CORPORATION (US) 2009-07-28 US disclosed
US-7566712-B2 Biaryl piperazinyl-pyridine analogues NEUROGEN CORPORATION (US) 2009-07-28 US disclosed