SCHEMBL3876977

SCHEMBL3876977

NC(=O)CNC(=O)Cc1cccc(Cl)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.58
KMT2A Q03164 3/20 0.58
MEN1 O00255 2/20 0.58
HPGD P15428 1/20 0.58
SMN1; SMN2 Q16637 1/20 0.58
MAPK8 P45983 1/20 0.54
HTR3E A5X5Y0 2/20 0.54
HTR3B O95264 2/20 0.54
HTR3A P46098 2/20 0.54
HTR3D Q70Z44 2/20 0.54
HTR3C Q8WXA8 2/20 0.54
EPHX2 P34913 2/20 0.54
SHMT1 P34896 1/20 0.53
SHMT2 P34897 1/20 0.53
NPC1 O15118 1/20 0.50
RAB9A P51151 1/20 0.50
KCNQ2 O43526 4/20 0.49
CTBP2 P56545 1/20 0.49
SIGMAR1 Q99720 1/20 0.47
HDAC3 O15379 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26423640 0.81 HTR3E (0.67) ALDH1A1KMT2AMEN1MAPK8HTR3E
SCHEMBL1395822 0.81 HTR3E (0.67) ALDH1A1KMT2AMEN1MAPK8HTR3E
SCHEMBL13181398 0.81 KMT2A (0.48) KMT2AHPGDSMN1; SMN2MAPK8SHMT1
SCHEMBL29481931 0.81 MEN1 (0.61) ALDH1A1KMT2AMEN1HPGDSMN1; SMN2
SCHEMBL17151448 0.81 MEN1 (0.61) ALDH1A1KMT2AMEN1HPGDSMN1; SMN2
SCHEMBL8858592 0.80 MEN1 (0.59) ALDH1A1KMT2AMEN1HPGDSMN1; SMN2
SCHEMBL924347 0.80 MEN1 (0.59) ALDH1A1KMT2AMEN1HPGDSMN1; SMN2
Hydrochloric Acid SCHEMBL2175078 0.80 HTR3E (0.65) ALDH1A1KMT2AMEN1MAPK8HTR3E
SCHEMBL7769258 0.80 KMT2A (0.57) ALDH1A1KMT2AMEN1HPGDEPHX2
SCHEMBL28992291 0.79 ALDH1A1 (0.68) ALDH1A1KMT2AMEN1HPGDSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1891064-B1 N-AMIDE DERIVATIVES OF 8-AZABICYCLO[3.2.1]OCT-3-YL AS CCR1 ANTAGONISTS ALMIRALL SA (ES) 2009-09-02 EP disclosed