SCHEMBL388066

SCHEMBL388066

O=CCNC(=O)c1ccc(-c2ccc(Cl)cc2)s1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESRRG P62508 6/20 0.59
ESR1 P03372 3/20 0.59
IKBKB O14920 1/20 0.55
MAPKAPK2 P49137 1/20 0.48
ESR2 Q92731 1/20 0.46
CNR1 P21554 1/20 0.46
RAB9A P51151 4/20 0.46
NPC1 O15118 3/20 0.46
PRSS12 P56730 1/20 0.46
PPARG P37231 1/20 0.46
NCOA2 Q15596 1/20 0.46
NCOA1 Q15788 1/20 0.46
NCOA3 Q9Y6Q9 1/20 0.46
HDAC1 Q13547 3/20 0.45
ACKR3 P25106 1/20 0.45
KDM4E B2RXH2 4/20 0.45
LMNA P02545 2/20 0.45
MAPT P10636 2/20 0.45
KMT2A Q03164 2/20 0.45
PTPN1 P18031 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20764262 0.78 ESRRG (0.78) ESRRGESR1IKBKBRAB9ANPC1
SCHEMBL8502506 0.75 IKBKB (0.65) ESRRGESR1IKBKBMAPKAPK2ESR2
SCHEMBL20764016 0.74 ESRRG (1.00) ESRRGESR1MAPKAPK2ESR2RAB9A
SCHEMBL20764080 0.73 ESRRG (0.78) ESRRGESR1MAPKAPK2ESR2CNR1
SCHEMBL1144473 0.73 IKBKB (0.71) ESRRGESR1IKBKBCNR1RAB9A
SCHEMBL5983409 0.73 IKBKB (0.71) ESRRGESR1IKBKBMAPKAPK2ESR2
SCHEMBL6378947 0.72 IKBKB (1.00) ESRRGESR1IKBKBMAPKAPK2ESR2
SCHEMBL4929313 0.71 AKT3 (0.62) CNR1RAB9ANPC1HDAC1ACKR3
SCHEMBL27677406 0.71 IKBKB (0.63) ESRRGESR1IKBKBCNR1RAB9A
SCHEMBL4930772 0.70 ESRRG (0.73) ESRRGESR1MAPKAPK2ESR2CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8101764-B2 MCH receptor antagonists ELI LILLY AND COMPANY (US) 2012-01-24 US disclosed