SCHEMBL3880682

SCHEMBL3880682

CC(=O)c1nc(-c2ccc(F)c(Cl)c2)cc(N2CCN(c3ncccc3C(F)(F)F)CC2)n1

nearest known ligand 0.46

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 8/20 0.46
TRPA1 O75762 1/20 0.46
TRPV1 Q8NER1 1/20 0.46
GAA P10253 1/20 0.45
RBP4 P02753 1/20 0.44
ALDH1A1 P00352 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3876557 0.92 GAA (0.47) HSD11B1TRPA1TRPV1GAARBP4
SCHEMBL3887718 0.90 GAA (0.46) HSD11B1TRPA1TRPV1GAAALDH1A1
SCHEMBL3885210 0.90 GAA (0.46) HSD11B1TRPA1TRPV1GAARBP4
SCHEMBL14614138 0.90 GAA (0.45) HSD11B1TRPA1TRPV1GAARBP4
SCHEMBL3878643 0.86 TRPA1 (0.43) HSD11B1TRPA1TRPV1GAARBP4
SCHEMBL3879411 0.86 TRPA1 (0.47) HSD11B1TRPA1TRPV1GAARBP4
SCHEMBL3877152 0.86 HSD11B1 (0.47) HSD11B1
SCHEMBL3875989 0.86 HSD11B1 (0.48) HSD11B1TRPA1TRPV1
SCHEMBL3880207 0.85 GALR2 (0.51) HSD11B1TRPV1
SCHEMBL3877637 0.85 HSD11B1 (0.46) HSD11B1GAARBP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7566712-B2 Biaryl piperazinyl-pyridine analogues NEUROGEN CORPORATION (US) 2009-07-28 US disclosed
US-7566712-B2 Biaryl piperazinyl-pyridine analogues NEUROGEN CORPORATION (US) 2009-07-28 US disclosed
US-7566712-B2 Biaryl piperazinyl-pyridine analogues NEUROGEN CORPORATION (US) 2009-07-28 US disclosed