SCHEMBL3884035

SCHEMBL3884035

CC(Cc1ccc(OC2Cc3ccccc3C2)c(-c2ccc3[nH]ncc3c2)c1)C(=O)O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 8/20 0.42
ROCK2 O75116 5/20 0.41
GSK3B P49841 3/20 0.41
CDK5 Q00535 3/20 0.41
DYRK1A Q13627 3/20 0.41
ROCK1 Q13464 3/20 0.41
AURKA O14965 2/20 0.41
CDK1 P06493 2/20 0.41
PRKACA P17612 2/20 0.41
RPS6KB1 P23443 2/20 0.41
CDK2 P24941 2/20 0.41
GSK3A P49840 2/20 0.41
CDC42BPA Q5VT25 2/20 0.41
AURKB Q96GD4 2/20 0.41
SGK2 Q9HBY8 2/20 0.41
DAPK3 O43293 1/20 0.41
JAK2 O60674 1/20 0.41
FGFR1 P11362 1/20 0.41
MARK3 P27448 1/20 0.41
MAPK1 P28482 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3891048 0.88 MAPK14 (0.41) TRPA1ROCK2GSK3BCDK5DYRK1A
SCHEMBL3881923 0.88 MAPK14 (0.40) TRPA1ROCK2GSK3BCDK5DYRK1A
SCHEMBL3889253 0.88 MAPK14 (0.40) TRPA1ROCK2GSK3BCDK5DYRK1A
SCHEMBL3888233 0.85 TRPA1 (0.40) TRPA1ROCK2GSK3BCDK5DYRK1A
SCHEMBL3882061 0.85 FFAR4 (0.45) TRPA1ROCK2GSK3BCDK5DYRK1A
SCHEMBL3895963 0.84 IKBKB (0.42) ROCK1AKT1PDE4APDE4BPDE4C
SCHEMBL3883918 0.83 TRPA1 (0.38) TRPA1ROCK2GSK3BCDK5DYRK1A
SCHEMBL3884504 0.83 AR (0.43) TRPA1PDE4APDE4BPDE4CPDE4D
SCHEMBL3884038 0.82 TRPA1 (0.42) TRPA1ROCK2PDE4APDE4BPDE4C
SCHEMBL3888551 0.81 FFAR4 (0.39) PDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1477472-B1 SUBSTITUTED PHENYLALKANOIC ACID DERIVATIVE AND USE THEREOF ASAHI KASEI PHARMA CORP (JP) 2009-01-14 EP claimed