SCHEMBL3885197

SCHEMBL3885197

CCC#CC(=O)C(C)NC(=O)O

nearest known ligand 0.34

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MME P08473 1/20 0.34
ACE P12821 1/20 0.34
CPA1 P15085 1/20 0.34
ACE2 Q9BYF1 1/20 0.34
CYP2D6 P10635 1/20 0.31
CYP2C19 P33261 1/20 0.31
GRIK1 P39086 1/20 0.30
GRIK2 Q13002 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4166454 0.77 CYP2D6 (0.30) CYP2D6CYP2C19
SCHEMBL26097761 0.77 CYP2D6 (0.30) CYP2D6CYP2C19
SCHEMBL4172764 0.75 CA1 (0.45) CYP2D6CYP2C19
SCHEMBL6957514 0.73
SCHEMBL17275451 0.70 CYP2D6 (0.31) CYP2D6CYP2C19
SCHEMBL22781615 0.68 EPHX1 (0.38)
SCHEMBL31036601 0.67 CYP2D6 (0.37) MMEACECPA1ACE2CYP2D6
SCHEMBL7088563 0.66 METAP2 (0.47)
SCHEMBL73409 0.65
SCHEMBL1152458 0.65

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2013184-A1 SULFONAMIDE COMPOUNDS USEFUL AS EDG RECEPTOR MODULATORS AstraZeneca AB (SE) 2009-01-14 EP disclosed
WO-2007129019-A1 SULFONAMIDE COMPOUNDS USEFUL AS EDG RECEPTOR MODULATORS ASTRAZENECA AB (SE) 2007-11-15 WO disclosed