SCHEMBL3887191

SCHEMBL3887191

O=C(O)CC(c1cnc2ccoc2c1)N1CCC(CCCc2ccc3c(n2)CCCN3)C1=O

nearest known ligand 0.63

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ITGAV P06756 20/20 0.63
ITGB3 P05106 19/20 0.63
ITGA2B P08514 4/20 0.41
ITGB6 P18564 3/20 0.40
ITGB1 P05556 3/20 0.40
ITGB8 P26012 2/20 0.40
ITGA5 P08648 2/20 0.40
ITGB5 P18084 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4045472 0.90 ITGAV (0.79) ITGAVITGB3ITGA2BITGB6ITGB1
SCHEMBL4047951 0.86 ITGAV (0.68) ITGAVITGB3ITGA2BITGB6ITGB1
SCHEMBL7556616 0.84 ITGAV (0.57) ITGAVITGB3ITGA2BITGB6ITGB1
SCHEMBL4371634 0.84 ITGAV (0.59) ITGAVITGB3ITGB6ITGB8
SCHEMBL3886608 0.83 ITGAV (0.57) ITGAVITGB3ITGA2BITGB6ITGB1
SCHEMBL4045463 0.80 ITGB3 (0.50) ITGAVITGB3ITGA2BITGB5
SCHEMBL7945748 0.79 ITGAV (0.77) ITGAVITGB3ITGA2BITGB6ITGB1
SCHEMBL7945753 0.79 ITGAV (0.77) ITGAVITGB3ITGA2BITGB6ITGB1
SCHEMBL7945568 0.78 ITGAV (1.00) ITGAVITGB3ITGA2BITGB6ITGB8
SCHEMBL3888492 0.78 ITGAV (1.00) ITGAVITGB3ITGA2BITGB6ITGB8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1047425-A4 INTEGRIN RECEPTOR ANTAGONISTS MERCK & CO INC (US) 2009-04-22 EP claimed
EP-1047425-A1 INTEGRIN RECEPTOR ANTAGONISTS Merck & Co., Inc. (US) 2000-11-02 EP claimed
WO-1999030709-A1 INTEGRIN RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 1999-06-24 WO claimed