SCHEMBL4047951

SCHEMBL4047951

O=C(O)CC(c1cnc2c(c1)OCC2)N1CCC(CCCc2ccc3c(n2)CCCN3)C1=O

nearest known ligand 0.68

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ITGAV P06756 20/20 0.68
ITGB3 P05106 19/20 0.68
ITGA2B P08514 6/20 0.40
ITGB6 P18564 3/20 0.40
ITGB8 P26012 2/20 0.40
ITGB1 P05556 2/20 0.40
ITGA5 P08648 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3888089 0.90 ITGAV (0.82) ITGAVITGB3ITGA2BITGB6ITGB8
SCHEMBL3887191 0.86 ITGAV (0.63) ITGAVITGB3ITGA2BITGB6ITGB8
SCHEMBL3886608 0.83 ITGAV (0.57) ITGAVITGB3ITGA2BITGB6ITGB8
SCHEMBL7944256 0.82 ITGAV (0.82) ITGAVITGB3ITGA2BITGB6ITGB8
SCHEMBL7944250 0.82 ITGAV (0.82) ITGAVITGB3ITGA2BITGB6ITGB8
SCHEMBL4371634 0.81 ITGAV (0.59) ITGAVITGB3ITGB6ITGB8
SCHEMBL3885043 0.81 ITGB3 (1.00) ITGAVITGB3ITGA2BITGB6ITGB1
SCHEMBL3886509 0.81 ITGB3 (1.00) ITGAVITGB3ITGA2BITGB6ITGB1
SCHEMBL3893571 0.81 ITGB3 (1.00) ITGAVITGB3ITGA2BITGB6ITGB1
SCHEMBL3885035 0.81 ITGB3 (1.00) ITGAVITGB3ITGA2BITGB6ITGB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1047425-A4 INTEGRIN RECEPTOR ANTAGONISTS MERCK & CO INC (US) 2009-04-22 EP disclosed
EP-1047425-A1 INTEGRIN RECEPTOR ANTAGONISTS Merck & Co., Inc. (US) 2000-11-02 EP disclosed
WO-1999030709-A1 INTEGRIN RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 1999-06-24 WO disclosed