SCHEMBL3887692

SCHEMBL3887692

NS(=O)(=O)N1CCc2c([nH]c3ccccc23)C1C(=O)O

nearest known ligand 0.56

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.56
MAPKAPK2 P49137 2/20 0.50
ABCG2 Q9UNQ0 7/20 0.49
ABCB1 P08183 4/20 0.49
ADRA1D P25100 1/20 0.49
ADRA1A P35348 1/20 0.49
ADRA1B P35368 1/20 0.49
SIRT1 Q96EB6 2/20 0.48
LMNA P02545 1/20 0.47
MMP2 P08253 1/20 0.47
PKM P14618 1/20 0.47
SIRT2 Q8IXJ6 1/20 0.46
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
MAPT P10636 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8111852 0.83 MMP2 (0.57) POLBMAPKAPK2ABCG2ABCB1ADRA1D
SCHEMBL8125346 0.82 MMP2 (0.56) POLBMAPKAPK2ABCG2ABCB1LMNA
SCHEMBL8123058 0.80 MMP2 (0.54) POLBMAPKAPK2ABCG2ABCB1ADRA1D
SCHEMBL8111675 0.80 MMP2 (0.54) POLBMAPKAPK2ABCG2ABCB1ADRA1D
SCHEMBL8121680 0.77 MMP2 (0.65) POLBMAPKAPK2ABCG2LMNAMMP2
SCHEMBL8129793 0.77 MMP2 (0.65) POLBMAPKAPK2ABCG2ABCB1LMNA
SCHEMBL9913669 0.77 ABCG2 (0.72) ABCG2ABCB1LMNAPKM
SCHEMBL8132615 0.76 MMP2 (0.58) POLBMAPKAPK2ABCG2ABCB1LMNA
SCHEMBL23438776 0.72 PKM (0.53) POLBABCG2ABCB1ADRA1DADRA1A
SCHEMBL6465789 0.72 ABCG2 (0.72) POLBABCG2ABCB1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1919475-B1 TETRAHYDRO- BETA-CARBOLIN-SULFONAMIDE DERIVATIVES AS 5-HT6 LIGANDS ESTEVE LABOR DR (ES) 2009-03-11 EP claimed