SCHEMBL3889347

SCHEMBL3889347

CC(=O)c1cc(C(=O)O)cc(C(=O)N[C@H](C)c2ccccc2)c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.57
LMNA P02545 4/20 0.57
NPC1 O15118 1/20 0.57
HDAC6 Q9UBN7 1/20 0.55
SMN1; SMN2 Q16637 2/20 0.54
MAPK1 P28482 2/20 0.52
ROCK2 O75116 1/20 0.52
RPS6KA5 O75582 1/20 0.52
MAP4K4 O95819 1/20 0.52
CDK1 P06493 1/20 0.52
CSF1R P07333 1/20 0.52
PRKACA P17612 1/20 0.52
FLT1 P17948 1/20 0.52
RPS6KB1 P23443 1/20 0.52
CDK2 P24941 1/20 0.52
AKT1 P31749 1/20 0.52
FLT4 P35916 1/20 0.52
KDR P35968 1/20 0.52
FLT3 P36888 1/20 0.52
GSK3A P49840 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3889350 1.00 ALDH1A1 (0.57) ALDH1A1LMNANPC1HDAC6SMN1; SMN2
SCHEMBL7948447 0.88 ALDH1A1 (0.57) ALDH1A1LMNANPC1SMN1; SMN2MAPK1
SCHEMBL3889792 0.87 NPC1 (0.61) ALDH1A1LMNANPC1SMN1; SMN2ROCK2
SCHEMBL3886906 0.87 ALDH1A1 (0.54) ALDH1A1LMNANPC1HDAC6SMN1; SMN2
SCHEMBL3886903 0.87 ALDH1A1 (0.54) ALDH1A1LMNANPC1HDAC6SMN1; SMN2
SCHEMBL7864711 0.87 NPC1 (0.61) ALDH1A1LMNANPC1SMN1; SMN2ROCK2
SCHEMBL13229354 0.87 GPR139 (0.64) ALDH1A1LMNANPC1SMN1; SMN2MAPK1
SCHEMBL27810867 0.87 ALDH1A1 (0.72) ALDH1A1LMNANPC1SMN1; SMN2MAPK1
SCHEMBL13229317 0.86 ALDH1A1 (0.52) ALDH1A1LMNANPC1SMN1; SMN2MAPK1
SCHEMBL13229107 0.84 ALDH1A1 (0.73) ALDH1A1LMNANPC1SMN1; SMN2MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7476764-B2 Phenylcarboxyamides as beta-secretase inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2009-01-13 US disclosed
US-7476764-B2 Phenylcarboxyamides as beta-secretase inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2009-01-13 US disclosed
US-7476764-B2 Phenylcarboxyamides as beta-secretase inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2009-01-13 US disclosed
US-20070032470-A1 Novel phenylcarboxyamides as beta-secretase inhibitors BRISTOL-MYERS SQUIBB COMPANY 2007-02-08 US disclosed
US-20070032470-A1 Novel phenylcarboxyamides as beta-secretase inhibitors BRISTOL-MYERS SQUIBB COMPANY 2007-02-08 US disclosed
US-20070032470-A1 Novel phenylcarboxyamides as beta-secretase inhibitors BRISTOL-MYERS SQUIBB COMPANY 2007-02-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070032470-A1 Novel phenylcarboxyamides as beta-secretase inhibitors BACE1, APP, BACE2 ALDH1A1 3847/4885LMNA 609/4885NPC1 553/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.