SCHEMBL3889496

SCHEMBL3889496

COOC(=O)c1cccnc1F

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAPRT Q6XQN6 1/20 0.58
TDP1 Q9NUW8 2/20 0.42
L3MBTL1 Q9Y468 7/20 0.41
NPC1 O15118 2/20 0.41
TSHR P16473 2/20 0.41
GLA P06280 1/20 0.41
LMNA P02545 2/20 0.40
POLB P06746 1/20 0.40
MAP2K1 Q02750 1/20 0.40
KMT2A Q03164 2/20 0.39
KDM4E B2RXH2 3/20 0.39
PKM P14618 1/20 0.38
ALDH1A1 P00352 3/20 0.38
MAPT P10636 2/20 0.38
CYP3A4 P08684 1/20 0.38
ALOX15 P16050 1/20 0.38
BLM P54132 1/20 0.38
AGER Q15109 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
ATM Q13315 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1807364 0.86 NAPRT (0.61) NAPRTTDP1L3MBTL1TSHRLMNA
SCHEMBL25421433 0.83 NAPRT (0.50) NAPRTTDP1L3MBTL1NPC1TSHR
SCHEMBL12897074 0.81 TSHR (0.59) NAPRTTDP1L3MBTL1NPC1TSHR
SCHEMBL5325713 0.79 LMNA (0.58) TDP1L3MBTL1LMNAPOLBKMT2A
SCHEMBL25421430 0.79 ALDH1A1 (0.62) NAPRTTDP1L3MBTL1NPC1TSHR
SCHEMBL9944381 0.78 NAPRT (0.56) NAPRTL3MBTL1NPC1LMNAPOLB
SCHEMBL16415899 0.78 NAPRT (0.56) NAPRTTDP1L3MBTL1NPC1TSHR
SCHEMBL13296381 0.76 TSHR (0.64) NAPRTTDP1L3MBTL1NPC1TSHR
SCHEMBL29195335 0.76 NAPRT (0.58) NAPRTTDP1L3MBTL1NPC1TSHR
SCHEMBL1811012 0.76 NAPRT (0.68) NAPRTTDP1L3MBTL1NPC1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010493-A2 PYRIDYL AMIDE T-TYPE CALCIUM CHANNEL ANTAGONISTS Merck & Co., Inc. (US) 2009-01-07 EP disclosed
WO-2007120729-A2 PYRIDYL AMIDE T-TYPE CALCIUM CHANNEL ANTAGONISTS MERCK & CO., INC. (US) 2007-10-25 WO disclosed