SCHEMBL3890376

SCHEMBL3890376

[C-]#[N+]Cc1ccc(Br)cc1

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 3/20 0.42
HTR2A P28223 1/20 0.42
CYP2A6 P11509 1/20 0.42
IDO1 P14902 4/20 0.41
PYCR1 P32322 2/20 0.34
ALDH1A1 P00352 3/20 0.33
ALOX15 P16050 2/20 0.33
AGER Q15109 1/20 0.33
MAPK1 P28482 1/20 0.33
APP P05067 1/20 0.33
KDM4E B2RXH2 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5672968 0.76 IDO1 (0.48) TAAR1IDO1
SCHEMBL2561988 0.75 TAAR1 (0.50) TAAR1HTR2ACYP2A6IDO1
SCHEMBL12374395 0.74 ALDH1A1 (0.50) ALDH1A1ALOX15MAPK1
SCHEMBL5183493 0.74 TAAR1 (0.42) TAAR1HTR2ACYP2A6IDO1PYCR1
SCHEMBL10204783 0.74 IDO1 (0.39) IDO1
SCHEMBL855864 0.74 TP53 (0.43) TAAR1CYP2A6IDO1ALDH1A1MAPK1
SCHEMBL3538182 0.74 IDO1 (0.46) TAAR1HTR2ACYP2A6IDO1ALDH1A1
SCHEMBL4890253 0.74 IDO1 (0.46) TAAR1CYP2A6IDO1ALDH1A1ALOX15
Hydrochloric Acid SCHEMBL3248101 0.72 TAAR1 (0.41) TAAR1HTR2ACYP2A6IDO1PYCR1
SCHEMBL1550703 0.72 TAAR1 (0.50) TAAR1IDO1PYCR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115611881-A Method for synthesizing novel VHL ligand 4-F-VH032 复旦大学 2023-01-17 CN claimed
CN-110520413-B Macrocyclic broad spectrum antibiotics 阿奇克斯制药公司 2023-02-17 CN disclosed
CN-115611881-A Method for synthesizing novel VHL ligand 4-F-VH032 复旦大学 2023-01-17 CN disclosed
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed
WO-2009145721-A1 ISOINDOLINE DERIVATIVES COMPRISING PHENYL GROUPS AND THEIR USE IN THE TREATMENT OF PAIN DISORDERS ASTRAZENECA AB (SE) 2009-12-03 WO disclosed
WO-2009145718-A1 ISOINDOLINE DERIVATIVES COMPRISING AN ADDITIONAL HETEROCYCLIC GROUP AND THEIR USE IN THE TREATMENT OF PAIN DISORDERS ASTRAZENECA AB (SE) 2009-12-03 WO disclosed