SCHEMBL3900469

SCHEMBL3900469

O=C(O)CCCC1CCC(c2ccc(Cl)cc2)CC1

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.49
FFAR4 Q5NUL3 1/20 0.46
CYP2C9 P11712 1/20 0.44
ESR2 Q92731 1/20 0.44
DGAT1 O75907 3/20 0.44
ALDH1A1 P00352 2/20 0.43
MAPT P10636 2/20 0.43
LMNA P02545 1/20 0.43
CHRM4 P08173 1/20 0.42
SOAT1 P35610 1/20 0.42
POLB P06746 1/20 0.42
DRD2 P14416 1/20 0.41
PTGDR2 Q9Y5Y4 1/20 0.41
LTA4H P09960 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4975059 1.00 IDO1 (0.49) IDO1FFAR4CYP2C9ESR2DGAT1
SCHEMBL5761802 0.86 IDO1 (0.46) IDO1FFAR4CYP2C9ESR2DGAT1
SCHEMBL4976344 0.86 IDO1 (0.46) IDO1FFAR4CYP2C9ESR2DGAT1
SCHEMBL27809490 0.83 IDO1 (0.49) IDO1CYP2C9ESR2DGAT1ALDH1A1
SCHEMBL28002072 0.81 IDO1 (0.61) IDO1DGAT1SOAT1
Bicarbonate SCHEMBL1719769 0.78 IDO1 (0.51) IDO1CYP2C9ALDH1A1MAPTLMNA
SCHEMBL8997300 0.78 DRD2 (0.54) IDO1CYP2C9ESR2ALDH1A1MAPT
SCHEMBL8997297 0.78 DRD2 (0.54) IDO1CYP2C9ESR2ALDH1A1MAPT
SCHEMBL12209860 0.77 AKR1C3 (0.50) FFAR4
SCHEMBL27616065 0.77 DRD2 (0.67) DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1646383-A4 DESIGN AND SYNTHESIS OF OPTIMIZED LIGANDS FOR PPAR BETHESDA PHARMACEUTICALS INC (US) 2009-03-25 EP disclosed
EP-1646383-A1 DESIGN AND SYNTHESIS OF OPTIMIZED LIGANDS FOR PPAR Bethesda Pharmaceuticals, Inc. (US) 2006-04-19 EP disclosed
WO-2005009437-A1 DESIGN AND SYNTHESIS OF OPTIMIZED LIGANDS FOR PPAR BETHESDA PHARMACEUTICALS, INC. (US) 2005-02-03 WO disclosed