SCHEMBL3901190

SCHEMBL3901190

Cc1cccc(C(CN)c2cccnc2)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 3/20 0.46
ROCK2 O75116 1/20 0.44
CFTR P13569 1/20 0.43
SLC6A2 P23975 1/20 0.43
SLC6A4 P31645 1/20 0.43
SLC6A3 Q01959 1/20 0.43
GOPC Q9HD26 1/20 0.43
AKT1 P31749 1/20 0.43
OPRM1 P35372 1/20 0.42
OPRD1 P41143 1/20 0.42
HTR2A P28223 1/20 0.41
TAAR1 Q96RJ0 1/20 0.41
CYP11B1 P15538 1/20 0.41
SMN1; SMN2 Q16637 3/20 0.41
PDE4D Q08499 1/20 0.40
KCNA5 P22460 3/20 0.40
CTSA P10619 1/20 0.40
LMNA P02545 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
KCNH2 Q12809 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4381016 0.85 TAAR1 (0.56) CYP19A1SLC6A2SLC6A4SLC6A3HTR2A
SCHEMBL4196224 0.85 CFTR (0.57) CYP19A1CFTRSLC6A2SLC6A4SLC6A3
SCHEMBL3910832 0.81 TAAR1 (0.64) CYP19A1SLC6A2SLC6A4SLC6A3HTR2A
SCHEMBL5307787 0.81 HTR2A (0.64) CFTRSLC6A2SLC6A4SLC6A3GOPC
SCHEMBL3911314 0.76 HTR2A (0.45) CYP19A1HTR2ATAAR1
SCHEMBL20773646 0.75 CTSA (0.47) CYP19A1CTSA
SCHEMBL1034162 0.74 HTR2A (0.68) CYP19A1CFTRSLC6A2SLC6A4SLC6A3
SCHEMBL3904458 0.74 SLC6A2 (0.47) CYP19A1SLC6A2SLC6A4SLC6A3HTR2A
SCHEMBL3282177 0.73 NOS1 (0.44) SLC6A2SLC6A4SLC6A3LMNAKCNH2
SCHEMBL3903975 0.72 CYP11B1 (0.44) CYP19A1CFTRSLC6A2SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2018364-A1 THERAPEUTIC FLUOROETHYL UREAS Allergan, Inc. (US) 2009-01-28 EP disclosed
WO-2007137029-A1 THERAPEUTIC FLUOROETHYL UREAS ALLERGAN, INC. (US) 2007-11-29 WO disclosed