SCHEMBL3904013

SCHEMBL3904013

CC[C@@H](C)[C@H](N)C(=O)N[C@@H](CC(C)C)C(=O)N[C@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H]([C]=O)CCC(=O)O

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERAP2 Q6P179 7/20 0.63
IL1RN P18510 6/20 0.57
ERAP1 Q9NZ08 5/20 0.57
EDNRA P25101 1/20 0.54
MMP2 P08253 7/20 0.53
MMP9 P14780 5/20 0.53
MMP8 P22894 5/20 0.53
MMP1 P03956 4/20 0.53
CTSC P53634 1/20 0.51
ECE1 P42892 2/20 0.50
ADAM10 O14672 1/20 0.50
ADAM12 O43184 1/20 0.50
ADAMTS4 O75173 1/20 0.50
MMP3 P08254 1/20 0.50
MMP7 P09237 1/20 0.50
MMP12 P39900 1/20 0.50
MMP13 P45452 1/20 0.50
MMP14 P50281 1/20 0.50
MMP15 P51511 1/20 0.50
MMP16 P51512 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3904009 1.00 ERAP2 (0.63) ERAP2IL1RNERAP1EDNRAMMP2
SCHEMBL2183714 0.94 ERAP2 (0.59) ERAP2IL1RNERAP1EDNRAMMP2
SCHEMBL27869302 0.88 ERAP2 (0.54) ERAP2IL1RNERAP1EDNRAMMP2
SCHEMBL16468411 0.87 CTSC (0.54) ERAP2MMP2MMP9MMP8MMP1
SCHEMBL3979342 0.87 ERAP2 (0.62) ERAP2IL1RNERAP1EDNRAMMP2
SCHEMBL30299207 0.86 ERAP2 (0.68) ERAP2IL1RNERAP1EDNRAMMP2
SCHEMBL29769026 0.86 ERAP2 (0.69) ERAP2IL1RNERAP1EDNRAECE1
SCHEMBL30051527 0.86 ECE1 (0.64) ERAP2IL1RNERAP1EDNRAMMP2
SCHEMBL2197039 0.84 ERAP2 (0.61) ERAP2IL1RNERAP1MMP2MMP9
SCHEMBL30918496 0.84 ERAP2 (0.63) ERAP2IL1RNERAP1EDNRAMMP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1906987-A4 METHODS AND COMPOSITIONS FOR EMERGENCY CONTRACEPTION USING ENDOTHELIN RECEPTOR ANTAGONISTS POPULATION COUNCIL INC (US) 2009-01-28 EP disclosed
EP-1906987-A1 METHODS AND COMPOSITIONS FOR EMERGENCY CONTRACEPTION USING ENDOTHELIN RECEPTOR ANTAGONISTS The Population Council, Inc. (US) 2008-04-09 EP disclosed
WO-2007012006-A1 METHODS AND COMPOSITIONS FOR EMERGENCY CONTRACEPTION USING ENDOTHELIN RECEPTOR ANTAGONISTS THE POPULATION COUNCIL, INC. (US) 2007-01-25 WO disclosed