SCHEMBL3914531

SCHEMBL3914531

COc1cc2c(Oc3ccc(NC(=O)c4nccn(Cc5ccccc5)c4=O)cc3F)ccnc2cc1OCCCN1CCOCC1

nearest known ligand 0.73

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MET P08581 19/20 0.73
FLT3 P36888 1/20 0.71
INSR P06213 1/20 0.70
KDR P35968 1/20 0.67

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3912896 0.92 MET (0.70) METFLT3INSRKDR
SCHEMBL30716533 0.90 MET (0.76) METFLT3INSRKDR
SCHEMBL6520309 0.88 MET (0.72) METFLT3INSRKDR
SCHEMBL198559 0.87 MET (0.70) METFLT3INSRKDR
SCHEMBL30716517 0.87 MET (0.72) METFLT3INSRKDR
SCHEMBL30716496 0.87 MET (0.71) METFLT3INSR
SCHEMBL3987180 0.87 MET (0.69) METFLT3INSRKDR
SCHEMBL30716518 0.87 MET (0.76) METFLT3INSR
SCHEMBL30716495 0.86 MET (0.76) METFLT3INSRKDR
SCHEMBL30716523 0.86 MET (0.70) METFLT3INSRKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110053931-A1 QUINOLINE COMPOUNDS AND METHODS OF USE GAUDINO JOHN 2011-03-03 US claimed
US-20110053931-A1 QUINOLINE COMPOUNDS AND METHODS OF USE GAUDINO JOHN 2011-03-03 US disclosed
US-20110053931-A1 QUINOLINE COMPOUNDS AND METHODS OF USE GAUDINO JOHN 2011-03-03 US disclosed
EP-2032538-A2 QUINOLINE COMPOUNDS AND METHODS OF USE Array Biopharma, Inc. (US) 2009-03-11 EP disclosed
WO-2007146824-A2 QUINOLINE COMPOUNDS AND METHODS OF USE ARRAY BIOPHARMA INC. (US) 2007-12-21 WO disclosed
WO-2007146824-A2 QUINOLINE COMPOUNDS AND METHODS OF USE ARRAY BIOPHARMA INC. (US) 2007-12-21 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110053931-A1 QUINOLINE COMPOUNDS AND METHODS OF USE TK1, ABL1, ROR1 MET 563/4885FLT3 49/4885INSR 390/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.