SCHEMBL3914919

SCHEMBL3914919

COc1cc2nccc(Oc3ccc(-c4ccc(NC(=O)c5ccc(F)cc5)c(=O)[nH]4)cc3F)c2cc1OC

nearest known ligand 0.56

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MET P08581 15/20 0.56
PDGFRA P16234 3/20 0.55
AXL P30530 5/20 0.54
KDR P35968 5/20 0.53
MST1R Q04912 2/20 0.52
KIT P10721 2/20 0.52
FLT4 P35916 1/20 0.52
FLT3 P36888 1/20 0.52
FGFR2 P21802 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3913675 0.82 MET (0.55) METPDGFRAAXLKDRMST1R
SCHEMBL3913677 0.77 MET (0.65) METAXL
SCHEMBL5824355 0.75 MET (0.70) METPDGFRAAXLKDRMST1R
SCHEMBL3921647 0.74 AXL (0.62) METPDGFRAAXLKDRKIT
SCHEMBL31412937 0.72 MET (0.60) METPDGFRAAXLKDRMST1R
SCHEMBL31412928 0.72 MET (0.75) METPDGFRAAXLKDRMST1R
SCHEMBL2860965 0.72 MET (0.63) METPDGFRAAXLKDRMST1R
SCHEMBL12635551 0.72 PDGFRA (0.78) METPDGFRAAXLKDRMST1R
SCHEMBL4401175 0.72 MET (0.76) METPDGFRAAXLKDRMST1R
SCHEMBL3794835 0.72 MET (0.59) METPDGFRAAXLKDRMST1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2032538-A2 QUINOLINE COMPOUNDS AND METHODS OF USE Array Biopharma, Inc. (US) 2009-03-11 EP disclosed
WO-2007146824-A2 QUINOLINE COMPOUNDS AND METHODS OF USE ARRAY BIOPHARMA INC. (US) 2007-12-21 WO disclosed