SCHEMBL3913675

SCHEMBL3913675

COc1cc2nccc(Oc3ccc(-c4cc[nH]c(=O)c4NC(=O)c4ccc(F)cc4)cc3F)c2cc1OC

nearest known ligand 0.55

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MET P08581 17/20 0.55
KDR P35968 4/20 0.54
MST1R Q04912 2/20 0.54
AXL P30530 5/20 0.53
KIT P10721 1/20 0.51
FLT4 P35916 1/20 0.51
FLT3 P36888 1/20 0.51
PDGFRA P16234 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3914919 0.82 MET (0.56) METKDRMST1RAXLKIT
SCHEMBL3913410 0.76 MET (0.61) METKDRMST1RAXLPDGFRA
SCHEMBL22923853 0.74 AXL (0.68) METKDRMST1RAXLKIT
SCHEMBL3922913 0.74 MET (0.64) METKDRMST1RAXL
SCHEMBL5824355 0.74 MET (0.70) METKDRMST1RAXLKIT
SCHEMBL3921647 0.74 AXL (0.62) METKDRAXLKITPDGFRA
SCHEMBL5301510 0.73 MET (0.44) METKDRAXL
SCHEMBL3913677 0.73 MET (0.65) METAXL
SCHEMBL31412937 0.72 MET (0.60) METKDRMST1RAXLKIT
SCHEMBL31412928 0.72 MET (0.75) METKDRMST1RAXLKIT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2032538-A2 QUINOLINE COMPOUNDS AND METHODS OF USE Array Biopharma, Inc. (US) 2009-03-11 EP disclosed
WO-2007146824-A2 QUINOLINE COMPOUNDS AND METHODS OF USE ARRAY BIOPHARMA INC. (US) 2007-12-21 WO disclosed