SCHEMBL3915944

SCHEMBL3915944

COc1cc(N)ccc1CN1CCN(S(C)(=O)=O)CC1

nearest known ligand 0.54

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 4/20 0.54
TSHR P16473 2/20 0.54
PDCD1 Q15116 1/20 0.53
CD274 Q9NZQ7 1/20 0.53
KDM4E B2RXH2 5/20 0.50
ALDH1A1 P00352 3/20 0.50
POLB P06746 1/20 0.50
HTT P42858 2/20 0.49
ALOX15 P16050 1/20 0.49
MAPK1 P28482 2/20 0.49
GAA P10253 1/20 0.49
MAPT P10636 1/20 0.49
KMT2A Q03164 3/20 0.48
MEN1 O00255 2/20 0.48
NPSR1 Q6W5P4 1/20 0.46
TP53 P04637 1/20 0.46
CYP3A4 P08684 1/20 0.43
HTR4 Q13639 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3997899 0.83 KDM4E (0.52) CYP2D6TSHRPDCD1CD274KDM4E
SCHEMBL2075627 0.82 NR1H2 (0.59) TSHRKDM4EALDH1A1POLBHTT
SCHEMBL22172136 0.82 GAA (0.56) CYP2D6TSHRKDM4EALDH1A1HTT
SCHEMBL30309437 0.82 GAA (0.56) CYP2D6TSHRKDM4EALDH1A1HTT
SCHEMBL2205074 0.82 TSHR (0.59) TSHRKDM4EALDH1A1HTTMAPK1
SCHEMBL3916828 0.81 ALDH1A1 (0.51) PDCD1CD274KDM4EALDH1A1POLB
SCHEMBL3179790 0.80 TSHR (0.59) TSHRKDM4EALDH1A1HTTMAPK1
SCHEMBL13861948 0.78 SMN1; SMN2 (0.48) KDM4EALDH1A1HTTALOX15MAPK1
SCHEMBL3919971 0.78 NR1H2 (0.70) CYP2D6KDM4EALDH1A1POLBHTT
SCHEMBL4263324 0.78 HTT (0.54) TSHRKDM4EALDH1A1HTTALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2038253-A1 BIPHENYL DERIVATIVES AND THEIR USE IN TREATING HEPATITIS C Arrow Therapeutics Limited (GB) 2009-03-25 EP disclosed
WO-2007138242-A1 BIPHENYL DERIVATIVES AND THEIR USE IN TREATING HEPATITIS C ARROW THERAPEUTICS LIMITED (GB) 2007-12-06 WO disclosed