SCHEMBL3997899

SCHEMBL3997899

COc1cc(C(N)=O)ccc1CN1CCN(S(C)(=O)=O)CC1

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.52
ALDH1A1 P00352 5/20 0.52
POLB P06746 1/20 0.52
ALOX15 P16050 1/20 0.51
HTT P42858 1/20 0.51
CYP2D6 P10635 2/20 0.50
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
TSHR P16473 1/20 0.50
PDCD1 Q15116 1/20 0.49
CD274 Q9NZQ7 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.47
LMNA P02545 1/20 0.44
OPRM1 P35372 1/20 0.44
MAPK1 P28482 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3841405 0.85 ALDH1A1 (0.51) KDM4EALDH1A1POLBCYP2D6MEN1
SCHEMBL16380640 0.85 MAPK1 (0.51) KDM4EALDH1A1POLBCYP2D6MEN1
SCHEMBL6947771 0.85 L3MBTL1 (0.59) KDM4EALDH1A1MEN1KMT2ATSHR
SCHEMBL4271324 0.84 L3MBTL1 (0.61) KDM4EALDH1A1POLBMEN1KMT2A
SCHEMBL3992921 0.83 IP6K1 (0.52) KDM4EALDH1A1ALOX15HTTOPRM1
SCHEMBL3915944 0.83 CYP2D6 (0.54) KDM4EALDH1A1POLBALOX15HTT
SCHEMBL4263319 0.81 CYP2D6 (0.52) KDM4EALDH1A1HTTCYP2D6MEN1
SCHEMBL3919981 0.80 NPSR1 (0.62) KDM4EALDH1A1ALOX15HTTCYP2D6
SCHEMBL2906362 0.77 KDM4E (0.60) KDM4EALDH1A1CYP2D6MEN1KMT2A
SCHEMBL2624464 0.73 L3MBTL1 (0.76) KDM4EALDH1A1HTTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2038253-A1 BIPHENYL DERIVATIVES AND THEIR USE IN TREATING HEPATITIS C Arrow Therapeutics Limited (GB) 2009-03-25 EP disclosed
WO-2007138242-A1 BIPHENYL DERIVATIVES AND THEIR USE IN TREATING HEPATITIS C ARROW THERAPEUTICS LIMITED (GB) 2007-12-06 WO disclosed