SCHEMBL3918072

SCHEMBL3918072

CCCC(OC(=O)c1ccncc1)[SiH](OC)OC

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 5/20 0.41
CYP1A2 P05177 2/20 0.41
CYP2C9 P11712 2/20 0.41
CYP2C19 P33261 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
NPC1 O15118 2/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
KMT2A Q03164 2/20 0.40
NFKB1 P19838 1/20 0.40
NFKB2 Q00653 1/20 0.40
RELA Q04206 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
HSD17B10 Q99714 1/20 0.39
ADRB2 P07550 1/20 0.37
ADRB1 P08588 1/20 0.37
ADRB3 P13945 1/20 0.37
NAPRT Q6XQN6 1/20 0.37
MAPT P10636 2/20 0.37
PRKCA P17252 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4350523 0.88 LMNA (0.43) LMNACYP1A2CYP2C9CYP2C19SMN1; SMN2
SCHEMBL3919137 0.87 KMT2A (0.42) LMNACYP1A2CYP2C9CYP2C19SMN1; SMN2
SCHEMBL962296 0.85 LMNA (0.46) LMNACYP1A2SMN1; SMN2NPC1CYP2D6
SCHEMBL3912018 0.81 CYP19A1 (0.52) LMNAMAPTMAPK1
SCHEMBL3910706 0.79 LMNA (0.47) LMNACYP1A2CYP2C9CYP2C19SMN1; SMN2
SCHEMBL3919092 0.77 KMT2A (0.43) LMNASMN1; SMN2NPC1KMT2ANAPRT
SCHEMBL3910933 0.75 KMT2A (0.44) LMNACYP1A2CYP2C9CYP2C19SMN1; SMN2
SCHEMBL11821905 0.75 LMNA (0.43) LMNACYP1A2CYP2C9CYP2C19SMN1; SMN2
SCHEMBL11821911 0.75 LMNA (0.43) LMNACYP1A2CYP2C9CYP2C19SMN1; SMN2
SCHEMBL3923456 0.72 KMT2A (0.46) LMNACYP1A2CYP2C9CYP2C19SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090277559-A1 METHOD FOR VULCANIZATION-ADHERING RUBBER COMPOSITION TO ADHERENT OF BRASS OR PLATED WITH BRASS, REINFORCING MEMBER FOR RUBBER ARTICLE, RUBBER-REINFORCING MEMBER COMPOSITE AND PNEUMATIC TIRE BRIDGESTONE CORPORATION (JP) 2009-11-12 US disclosed
EP-1840158-B1 METHOD FOR VULCANIZATION AND ADHESION OF RUBBER COMPOSITION WITH ARTICLE TO BE ADHERED BEING MADE OF BRASS OR PLATED WITH BRASS, REINFORCING MATERIAL FOR RUBBER ARTICLE, RUBBER-REINFORCING MATERIAL COMPOSITE, AND PNEUMATIC TIRE BRIDGESTONE CORP (JP) 2009-02-18 EP disclosed
EP-1840158-A1 METHOD FOR VULCANIZATION AND ADHESION OF RUBBER COMPOSITION WITH ARTICLE TO BE ADHERED BEING MADE OF BRASS OR PLATED WITH BRASS, REINFORCING MATERIAL FOR RUBBER ARTICLE, RUBBER-REINFORCING MATERIAL COMPOSITE, AND PNEUMATIC TIRE Bridgestone Corporation (JP) 2007-10-03 EP disclosed