SCHEMBL3923919

SCHEMBL3923919

CCCCCc1c(C)coc1C

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.35
ALDH1A1 P00352 2/20 0.34
ALDH1A2 O94788 1/20 0.34
ALDH2 P05091 1/20 0.34
ALDH1B1 P30837 1/20 0.34
ALDH1A3 P47895 1/20 0.34
PTGS2 P35354 4/20 0.33
CYP3A4 P08684 2/20 0.33
CYP19A1 P11511 1/20 0.33
MAPT P10636 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
CCR5 P51681 2/20 0.33
ALOX5 P09917 1/20 0.33
ESR1 P03372 2/20 0.32
ADRA2A P08913 2/20 0.32
ADORA3 P0DMS8 2/20 0.32
TACR2 P21452 2/20 0.32
SLC6A2 P23975 2/20 0.32
SLC6A4 P31645 2/20 0.32
SLC6A3 Q01959 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3929292 0.93 NPC1 (0.38) THRBALDH1A1ALDH1A2ALDH2ALDH1B1
SCHEMBL3923923 0.86 ALDH1A1 (0.39) ALDH1A1ALDH1A2ALDH2ALDH1B1ALDH1A3
SCHEMBL16701741 0.72 TYR (0.42) ALDH1A1PTGS2CYP3A4MAPTSMN1; SMN2
SCHEMBL3930085 0.72 MAPT (0.36) ALDH1A1ALDH1A2ALDH2ALDH1B1ALDH1A3
SCHEMBL3920357 0.72 TYR (0.34) THRBALDH1A1ALDH1A2ALDH2ALDH1B1
SCHEMBL3922014 0.71 TYR (0.37) THRBALDH1A1ALDH1A2ALDH2ALDH1B1
SCHEMBL14389463 0.71 MAPT (0.35) ALDH1A1ALDH1A2ALDH2ALDH1B1ALDH1A3
SCHEMBL3918783 0.71 TYR (0.37) THRBALDH1A1ALDH1A2ALDH2ALDH1B1
SCHEMBL5679424 0.69 TSHR (0.50) THRBALDH1A1PTGS2CYP3A4CYP19A1
SCHEMBL11619551 0.67 TYR (0.38) ALDH1A1PTGS2CYP3A4MAPTALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2027101-A1 TRISUBSTITUTED FURAN DERIVATIVES AS FRAGRANCES AND AROMA SUBSTANCES Symrise GmbH & Co. KG (DE) 2009-02-25 EP disclosed
WO-2007131834-A1 TRISUBSTITUTED FURAN DERIVATIVES AS FRAGRANCES AND AROMA SUBSTANCES SYMRISE GMBH & CO. KG (DE) 2007-11-22 WO disclosed