SCHEMBL3931024

SCHEMBL3931024

O=C(O)CCCc1ccc(Cl)cn1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXRA P19793 2/20 0.46
RXRB P28702 2/20 0.46
RXRG P48443 2/20 0.46
FFAR1 O14842 1/20 0.45
SMN1; SMN2 Q16637 2/20 0.43
MAPK1 P28482 2/20 0.43
HDAC3 O15379 1/20 0.43
ADRA1A P35348 1/20 0.43
HDAC4 P56524 1/20 0.43
SLC6A3 Q01959 1/20 0.43
HDAC1 Q13547 1/20 0.43
HDAC7 Q8WUI4 1/20 0.43
HDAC2 Q92769 1/20 0.43
HDAC10 Q969S8 1/20 0.43
HDAC11 Q96DB2 1/20 0.43
HDAC8 Q9BY41 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
HDAC9 Q9UKV0 1/20 0.43
HDAC5 Q9UQL6 1/20 0.43
ALDH1A1 P00352 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24867307 0.89 FFAR1 (0.55) RXRARXRBRXRGFFAR1HDAC6
SCHEMBL11656517 0.81 HDAC3 (0.53) RXRARXRBRXRGFFAR1SMN1; SMN2
SCHEMBL7206139 0.79 SMN1; SMN2 (0.47) RXRARXRBRXRGFFAR1SMN1; SMN2
SCHEMBL15270538 0.79 TSHR (0.50) FFAR1SMN1; SMN2MAPK1HDAC3ADRA1A
SCHEMBL9655945 0.79 FFAR1 (0.45) FFAR1SMN1; SMN2MAPK1HDAC3ADRA1A
SCHEMBL3937280 0.79 FFAR1 (0.45) RXRARXRBRXRGFFAR1SMN1; SMN2
SCHEMBL3931150 0.79 NPSR1 (0.44) SMN1; SMN2MAPK1ALDH1A1POLBL3MBTL1
SCHEMBL29594052 0.79 SMN1; SMN2 (0.62) SMN1; SMN2MAPK1HDAC1HDAC2ALDH1A1
SCHEMBL12984996 0.78 L3MBTL1 (0.44) L3MBTL1LMNATSHRNPC1PLAU
SCHEMBL9656043 0.77 TBXAS1 (0.51) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009007418-A1 NOVEL BRONCHODILATING ISOQUINOLINE AMIDES RESPIRATORIUS AB (SE) 2009-01-15 WO disclosed
WO-2009007418-A1 NOVEL BRONCHODILATING ISOQUINOLINE AMIDES RESPIRATORIUS AB (SE) 2009-01-15 WO disclosed