SCHEMBL3932038

SCHEMBL3932038

COc1ccc2c(c1)c(=O)oc(=O)n2Cc1ccc(F)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.56
TSHR P16473 2/20 0.56
LMNA P02545 1/20 0.56
CYP1A2 P05177 1/20 0.56
CYP3A4 P08684 1/20 0.56
CYP2C9 P11712 1/20 0.56
CYP2C19 P33261 1/20 0.56
BLM P54132 1/20 0.56
PMP22 Q01453 1/20 0.56
NPSR1 Q6W5P4 1/20 0.56
KMT2A Q03164 2/20 0.51
RXFP1 Q9HBX9 2/20 0.48
TNIK Q9UKE5 1/20 0.48
PIK3R1 P27986 1/20 0.47
PIK3CA P42336 1/20 0.47
DRD2 P14416 1/20 0.47
DRD4 P21917 1/20 0.47
DRD3 P35462 1/20 0.47
PTGS1 P23219 1/20 0.47
PTGS2 P35354 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3932904 0.86 IDO1 (0.57) KMT2ATNIKPOLBIDO1CD74
SCHEMBL30908758 0.84 IDO1 (0.51) TSHRLMNACYP1A2CYP3A4CYP2C9
SCHEMBL606151 0.84 IDO1 (0.51) TSHRLMNACYP1A2CYP3A4CYP2C9
SCHEMBL3929699 0.82 IDO1 (0.60) KMT2ATNIKPOLBIDO1CD74
SCHEMBL2859999 0.80 KDM4E (0.53) KDM4ETSHRLMNARXFP1MAPK1
SCHEMBL2860677 0.80 P2RX4 (0.68) KMT2AMAPK1POLBIDO1TP53
SCHEMBL3921896 0.79 KMT2A (0.54) KMT2ATNIKPOLBIDO1CD74
SCHEMBL5123471 0.78 MIF (0.67) KDM4EKMT2ATNIKPOLBIDO1
SCHEMBL9046095 0.78 PLA2G2A (0.46) TSHRLMNACYP1A2CYP3A4CYP2C9
SCHEMBL368418 0.78 MIF (0.55) TSHRLMNANPSR1KMT2ATNIK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1786807-B1 HETEROCYCLIC ANTIVIRAL COMPOUNDS HOFFMANN LA ROCHE (CH) 2009-07-29 EP disclosed
US-7479489-B2 Heterocyclic antiviral compounds ROCHE PALO ALTO LLC (US) 2009-01-20 US disclosed
US-20060040927-A1 Heterocyclic antiviral compounds ROCHE PALO ALTO LLC 2006-02-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060040927-A1 Heterocyclic antiviral compounds HAVCR2, POLR1A, HCCS KDM4E 2915/4885TSHR 2710/4885LMNA 2439/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.