SCHEMBL30908758

SCHEMBL30908758

COc1ccc(Cn2c(=O)oc(=O)c3cc(Cl)ccc32)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 4/20 0.51
CCR2 P41597 1/20 0.51
P2RX4 Q99571 1/20 0.50
PTGS1 P23219 1/20 0.47
PTGS2 P35354 1/20 0.47
MAPT P10636 2/20 0.47
MEN1 O00255 1/20 0.47
RGS12 O14924 1/20 0.47
ALDH1A1 P00352 1/20 0.47
LMNA P02545 1/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2C9 P11712 1/20 0.47
PKM P14618 1/20 0.47
TSHR P16473 1/20 0.47
NFKB1 P19838 1/20 0.47
MAPK1 P28482 1/20 0.47
CYP2C19 P33261 1/20 0.47
GNAI1 P63096 1/20 0.47
PMP22 Q01453 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL606151 1.00 IDO1 (0.51) IDO1CCR2P2RX4PTGS1PTGS2
SCHEMBL10036738 0.86 IDO1 (0.55) IDO1P2RX4PTGS2MEN1ALDH1A1
SCHEMBL3932038 0.84 KDM4E (0.56) IDO1P2RX4PTGS1PTGS2MAPT
SCHEMBL2859999 0.84 KDM4E (0.53) P2RX4MAPTALDH1A1LMNATSHR
SCHEMBL9046095 0.83 PLA2G2A (0.46) PTGS1PTGS2MAPTMEN1RGS12
SCHEMBL2860677 0.83 P2RX4 (0.68) IDO1P2RX4MEN1ALDH1A1MAPK1
SCHEMBL3929699 0.83 IDO1 (0.60) IDO1ALDH1A1KMT2APOLBCD74
SCHEMBL5535346 0.83 IDO1 (0.54) IDO1P2RX4MAPTKMT2APOLB
SCHEMBL31019833 0.82 CCR2 (0.58) CCR2P2RX4PTGS1PTGS2MAPT
SCHEMBL4847252 0.80 PDE1B (0.47) MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118055923-A Benzodiazepine derivatives as positive allosteric modulators of the GABAA γ1 receptor 豪夫迈·罗氏有限公司 2024-05-17 CN disclosed