SCHEMBL3934985

SCHEMBL3934985

Cc1cc(Br)c2nc(Cl)ccc2c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 2/20 0.41
CCR5 P51681 2/20 0.41
CCR8 P51685 2/20 0.41
CYP1A2 P05177 3/20 0.34
CYP2A6 P11509 2/20 0.34
PRNP P04156 2/20 0.33
NPSR1 Q6W5P4 2/20 0.33
PSMD14 O00487 1/20 0.33
COPS5 Q92905 1/20 0.33
LMNA P02545 1/20 0.33
HPGD P15428 1/20 0.33
HTT P42858 1/20 0.33
NOD2 Q9HC29 1/20 0.33
BACE1 P56817 2/20 0.32
NQO2 P16083 2/20 0.32
NCK1 P16333 1/20 0.32
MAPT P10636 2/20 0.32
RXFP1 Q9HBX9 2/20 0.32
KDM4E B2RXH2 1/20 0.32
PPARG P37231 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31627462 0.80 CCR1 (0.43) CCR1CCR5CCR8CYP1A2CYP2A6
SCHEMBL20660798 0.78 BACE1 (0.33) CYP1A2CYP2A6BACE1MAPTRXFP1
SCHEMBL9088995 0.77 CCR1 (0.41) CCR1CCR5CCR8CYP1A2CYP2A6
SCHEMBL17582675 0.74 PRNP (0.44) CCR1CCR5CCR8CYP1A2CYP2A6
SCHEMBL7264434 0.73 NQO2 (0.44) CCR1CCR5CCR8CYP2A6PRNP
SCHEMBL20660923 0.73 BACE1 (0.38) BACE1
SCHEMBL30908523 0.72 POLB (0.37) LMNABACE1MAPTKDM4ESMN1; SMN2
SCHEMBL15448465 0.72 POLB (0.37) LMNABACE1MAPTKDM4ESMN1; SMN2
SCHEMBL31219687 0.72 ALDH1A1 (0.36) CCR1CCR5CCR8PRNPNPSR1
SCHEMBL3927988 0.72 LMNA (0.36) CCR1CCR5CCR8CYP1A2CYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090018163-A1 Substituted Heterocyclic Ethers and Their Use in CNS Disorders BRISTOL-MYERS SQUIBB COMPANY 2009-01-15 US disclosed
US-20090018163-A1 Substituted Heterocyclic Ethers and Their Use in CNS Disorders BRISTOL-MYERS SQUIBB COMPANY 2009-01-15 US disclosed
US-20090018163-A1 Substituted Heterocyclic Ethers and Their Use in CNS Disorders BRISTOL-MYERS SQUIBB COMPANY 2009-01-15 US disclosed
WO-2009009633-A1 SUBSTITUTED HETEROCYCLIC ETHERS AND THEIR USE IN CNS DISORDERS BRISTOL-MYERS SQUIBB COMPANY (US) 2009-01-15 WO disclosed
US-5491126-A BENZOTRIAZINE DERIVATIVES E. I. DU PONT DE NEMOURS AND COMPANY (US) 1996-02-13 US disclosed
US-5389600-A A phenyl quinoxaline or benzotriazine antigrowth agents E. I. DU PONT DE NEMOURS AND COMPANY (US) 1995-02-14 US disclosed
EP-0559843-B1 SUBSTITUTED N-HETEROBICYCLIC HERBICIDES DU PONT (US) 1994-09-14 EP disclosed
EP-0559843-A1 SUBSTITUTED N-HETEROBICYCLIC HERBICIDES. DU PONT (US) 1993-09-15 EP disclosed
WO-1992009578-A1 SUBSTITUTED FUSED HETEROCYCLIC HERBICIDES E.I. DU PONT DE NEMOURS AND COMPANY (US) 1992-06-11 WO disclosed
US-5110347-A Pre- and postemergence; quinoxaline derivatives E. I DU PONT DE NEMOURS AND COMPANY (US) 1992-05-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090018163-A1 Substituted Heterocyclic Ethers and Their Use in CNS Disorders CNR1, CNR2, PMP22 CCR1 736/4885CCR5 1343/4885CCR8 1009/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.