SCHEMBL3935675

SCHEMBL3935675

COc1cc(Cl)cc(CCc2cc(N)n[nH]2)c1

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
FGFR2 P21802 13/20 0.44
FGFR1 P11362 10/20 0.44
FGFR3 P22607 7/20 0.44
DYRK1A Q13627 1/20 0.42
CYP19A1 P11511 1/20 0.42
DAO P14920 1/20 0.40
FGFR4 P22455 2/20 0.37
LTA4H P09960 1/20 0.37
KDR P35968 4/20 0.36
AURKA O14965 1/20 0.36
JAK2 O60674 1/20 0.36
PDGFRB P09619 1/20 0.36
FLT3 P36888 1/20 0.36
IGF1R P08069 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1922681 0.90 CYP19A1 (0.51) FGFR2FGFR1FGFR3DYRK1ACYP19A1
SCHEMBL4016450 0.80 DYRK1A (0.58) FGFR2FGFR1FGFR3DYRK1ACYP19A1
SCHEMBL3940159 0.79 DYRK1A (0.43) FGFR2FGFR1FGFR3DYRK1ACYP19A1
SCHEMBL4012249 0.79 TAAR1 (0.54) FGFR2FGFR1FGFR3DYRK1ADAO
SCHEMBL4016522 0.77 DYRK1A (0.40) FGFR2FGFR1FGFR3DYRK1ACYP19A1
SCHEMBL4012062 0.76 FGFR3 (0.44) FGFR2FGFR1FGFR3DYRK1ADAO
SCHEMBL17967278 0.74 MKNK1 (0.54) DAOLTA4H
SCHEMBL23409093 0.73 FGFR2 (0.52) FGFR2FGFR1FGFR3CYP19A1DAO
SCHEMBL5103566 0.72 FGFR1 (0.59) FGFR2FGFR1FGFR3KDRIGF1R
SCHEMBL5281973 0.72 TAAR1 (0.55) CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2044063-A1 PYRIMIDINE DERIVATIVES USEFUL IN THE TREATMENT OF CANCER Astra Zeneca AB (SE) 2009-04-08 EP disclosed
WO-2008001070-A1 PYRIMIDINE DERIVATIVES USEFUL IN THE TREATMENT OF CANCER ASTRAZENECA AB (SE) 2008-01-03 WO disclosed
US-20080004302-A1 Novel Compounds ASTRAZENECA AB (SE) 2008-01-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080004302-A1 Novel Compounds CYP11B2, CYP11B1, CYP46A1 FGFR2 2044/4885FGFR1 1428/4885FGFR3 2897/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.