SCHEMBL3936032

SCHEMBL3936032

O=C(Nc1ccc(Cl)c(C(=O)Nc2cccnc2)c1)c1cc(N2CCOCC2)cc(C(F)(F)F)c1

nearest known ligand 0.66

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CSF1R P07333 12/20 0.66
MAPK14 Q16539 2/20 0.56
MAPK13 O15264 1/20 0.56
MAPK12 P53778 1/20 0.56
MAPK11 Q15759 1/20 0.56
SMN1; SMN2 Q16637 2/20 0.54
MEN1 O00255 1/20 0.54
KMT2A Q03164 1/20 0.54
BRAF P15056 4/20 0.53
RAF1 P04049 2/20 0.53
TP53 P04637 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3929957 0.82 CSF1R (0.78) CSF1RMAPK14BRAF
SCHEMBL1276893 0.80 CSF1R (1.00) CSF1RMAPK14MEN1KMT2ABRAF
SCHEMBL1420016 0.79 RAF1 (0.65) CSF1RBRAFRAF1
SCHEMBL3933053 0.76 SMN1; SMN2 (0.60) CSF1RMAPK14SMN1; SMN2MEN1KMT2A
SCHEMBL3934404 0.75 CSF1R (0.83) CSF1RBRAF
SCHEMBL3934946 0.74 CSF1R (0.60) CSF1RSMN1; SMN2MEN1KMT2ABRAF
SCHEMBL13459839 0.74 RAF1 (0.52) CSF1RMAPK14SMN1; SMN2BRAFRAF1
SCHEMBL5487784 0.74 CSF1R (0.55) CSF1RBRAFRAF1
SCHEMBL22772386 0.74 ABL1 (0.63) CSF1RMAPK14BRAFRAF1
SCHEMBL3944484 0.74 CSF1R (0.73) CSF1RMAPK14BRAF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1831198-B1 PYRIDINE CARBOXAMIDE DERIVATIVES FOR USE AS ANTICANCER AGENTS ASTRAZENECA AB (SE) 2009-04-08 EP disclosed