SCHEMBL3936147

SCHEMBL3936147

Cc1cc(Nc2nc(Cl)nc(N3CCOCC3)n2)n[nH]1

nearest known ligand 0.60

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 1/20 0.60
AURKA O14965 4/20 0.52
AURKB Q96GD4 1/20 0.52
TDP1 Q9NUW8 1/20 0.50
JAK2 O60674 5/20 0.49
JAK3 P52333 5/20 0.49
MAPT P10636 1/20 0.47
LMNA P02545 1/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
IGF1R P08069 1/20 0.47
PTGS2 P35354 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10294568 0.87 AURKA (0.56) AURKAAURKB
SCHEMBL3005925 0.83 IGF1R (0.59) IGF1R
SCHEMBL3936381 0.82 TDP1 (0.51) NTRK1TDP1MAPTLMNACYP1A2
SCHEMBL3939475 0.79 PAK4 (0.56) NTRK1AURKAAURKBJAK2JAK3
SCHEMBL10312104 0.78 NTRK1 (0.54) NTRK1AURKAAURKBTDP1JAK2
SCHEMBL219543 0.78 JAK3 (0.59) NTRK1AURKAAURKBJAK2JAK3
SCHEMBL10312145 0.78 AURKA (0.56) NTRK1AURKAAURKBJAK2JAK3
SCHEMBL13943376 0.76 JAK3 (0.76) NTRK1AURKAAURKBJAK2JAK3
SCHEMBL23321312 0.75 LMNA (0.82) TDP1MAPTLMNACYP1A2CYP3A4
SCHEMBL10312220 0.74 NTRK1 (0.50) NTRK1AURKAAURKBJAK2JAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009016410-A2 CHEMICAL COMPOUNDS 831 ASTRAZENECA AB (SE) 2009-02-05 WO disclosed