SCHEMBL3937389

SCHEMBL3937389

CC(C)(C)OC(=O)N1CCC(COCCc2cc(Cl)cc3cn(CC4CC4)nc23)(c2ccc(F)cc2)CC1

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 7/20 0.40
SLC6A4 P31645 6/20 0.37
KCNH2 Q12809 6/20 0.37
CCR5 P51681 5/20 0.37
CNR2 P34972 2/20 0.36
CNR1 P21554 1/20 0.36
JAK2 O60674 2/20 0.35
JAK1 P23458 2/20 0.35
PDE4A P27815 1/20 0.35
PDE4B Q07343 1/20 0.35
PDE4C Q08493 1/20 0.35
PDE4D Q08499 1/20 0.35
BACE1 P56817 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3935761 0.89 JAK2 (0.40) TACR1SLC6A4KCNH2JAK2JAK1
SCHEMBL3937761 0.85 TACR1 (0.38) TACR1SLC6A4KCNH2CCR5CNR2
SCHEMBL2427977 0.84 CCR5 (0.37) TACR1CCR5CNR2CNR1JAK2
SCHEMBL2427974 0.84 CCR5 (0.37) TACR1CCR5CNR2CNR1JAK2
SCHEMBL3928416 0.83 TACR1 (0.37) TACR1SLC6A4KCNH2CCR5
SCHEMBL3934912 0.83 TACR1 (0.42) TACR1SLC6A4KCNH2CCR5CNR2
SCHEMBL3935027 0.80 TACR1 (0.38) TACR1SLC6A4KCNH2
SCHEMBL3924880 0.79 ACACB (0.46) TACR1SLC6A4KCNH2CCR5
SCHEMBL3938855 0.79 TACR1 (0.36) TACR1SLC6A4KCNH2
SCHEMBL3935765 0.79 TACR1 (0.47) TACR1SLC6A4KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009009411-A1 SUBSTITUTED HETEROCYCLIC ETHERS AND THEIR USE IN CNS DISORDERS BRISTOL-MYERS SQUIBB COMPANY (US) 2009-01-15 WO disclosed