SCHEMBL3940196

SCHEMBL3940196

CCc1c(C(=O)Nc2ccc3c(c2)CCNC3)nnn1Cc1ccc(Cl)c(Cl)c1

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 2/20 0.43
NPC1 O15118 4/20 0.42
RAB9A P51151 4/20 0.42
KDM4E B2RXH2 1/20 0.41
MAPK1 P28482 1/20 0.41
USP28 Q96RU2 1/20 0.41
PTGDR2 Q9Y5Y4 1/20 0.41
SLC2A1 P11166 1/20 0.40
F2 P00734 1/20 0.40
PLG P00747 1/20 0.40
PLAU P00749 1/20 0.40
PLAT P00750 1/20 0.40
KLKB1 P03952 1/20 0.40
PRSS1 P07477 1/20 0.40
BLM P54132 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
MAPT P10636 1/20 0.39
MELK Q14680 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3939653 0.99 S1PR1 (0.42) S1PR1NPC1RAB9AKDM4EMAPK1
SCHEMBL13944421 0.81 THRB (0.51) NPC1RAB9AKDM4ESMN1; SMN2MAPT
SCHEMBL13943968 0.80 MAPT (0.48) S1PR1USP28SLC2A1F2PLG
SCHEMBL3611038 0.79 PTGDR2 (0.47) RAB9AUSP28PTGDR2SLC2A1F2
SCHEMBL3942819 0.79 SLC2A1 (0.45) S1PR1NPC1RAB9AKDM4ESLC2A1
Hydrochloric Acid SCHEMBL3602662 0.79 PTGDR2 (0.47) RAB9AUSP28PTGDR2SLC2A1F2
Hydrochloric Acid SCHEMBL3946111 0.78 SLC2A1 (0.46) S1PR1NPC1RAB9AKDM4ESLC2A1
SCHEMBL3943729 0.78 MELK (0.44) S1PR1NPC1RAB9AKDM4EMAPK1
SCHEMBL13504961 0.77 USP28 (0.44) USP28PTGDR2SLC2A1F2PLG
Hydrochloric Acid SCHEMBL3948321 0.77 MELK (0.43) S1PR1NPC1RAB9AKDM4EMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009016216-A1 TRIAZOLE DERIVATIVES AS SCD INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2009-02-05 WO claimed
WO-2009016216-A1 TRIAZOLE DERIVATIVES AS SCD INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2009-02-05 WO disclosed