SCHEMBL3940281

SCHEMBL3940281

COC(=O)N(Cc1ccc(C(=O)Nc2ccccc2N)cc1)c1cccnc1.CS(=O)(=O)O

nearest known ligand 0.55

Known targets — ChEMBL curated mechanism

ABL1ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB2AGTR1BCL2BCL2A1BCL2L1BCL2L10BCL2L2BCRBRAFCHRM1CHRNA10CHRNA9DRD1DRD2DRD3DRD4DRD5EGFRF2FLT1FLT4GCKGHSRGNRHRGRIN1GRIN2AGRIN2BGRIN2CGRIN2DGRIN3AGRIN3BHTR1AHTR1BHTR1DHTR2AHTR2CHTR3AIDH2KDRKITMAOBMCL1MTTPPP4HBPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PIKFYVEROCK1ROCK2SLC18A2SLC6A2SLC6A3SLC6A4TACR1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8gyrAgyrBparCparEpol

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 19/20 0.55
HDAC3 O15379 6/20 0.55
HDAC2 Q92769 6/20 0.55
NCOR2 Q9Y618 4/20 0.55
HDAC11 Q96DB2 4/20 0.52
HDAC8 Q9BY41 4/20 0.52
HDAC6 Q9UBN7 4/20 0.52
HDAC4 P56524 3/20 0.52
HDAC7 Q8WUI4 3/20 0.52
HDAC10 Q969S8 3/20 0.52
HDAC9 Q9UKV0 3/20 0.52
HDAC5 Q9UQL6 3/20 0.52
CYP3A4 P08684 2/20 0.52
KDM1A O60341 1/20 0.52
F3 P13726 1/20 0.52
NAMPT P43490 2/20 0.49
NCOR1 O75376 1/20 0.48
GAA P10253 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Sulfuric Acid SCHEMBL3948204 0.98 HDAC1 (0.55) HDAC1HDAC3HDAC2NCOR2HDAC11
SCHEMBL30006351 0.96 HDAC1 (0.59) HDAC1HDAC3HDAC2NCOR2HDAC11
SCHEMBL2175904 0.96 HDAC1 (0.59) HDAC1HDAC3HDAC2NCOR2HDAC11
Hydrochloric Acid SCHEMBL3943756 0.95 HDAC1 (0.58) HDAC1HDAC3HDAC2NCOR2HDAC11
Bromide SCHEMBL3943842 0.95 HDAC1 (0.58) HDAC1HDAC3HDAC2NCOR2HDAC11
Acetic Acid SCHEMBL4103112 0.94 HDAC1 (0.59) HDAC1HDAC3HDAC2NCOR2HDAC11
Phosphoric Acid SCHEMBL3948469 0.94 HDAC1 (0.56) HDAC1HDAC3HDAC2NCOR2HDAC11
SCHEMBL3941359 0.92 HDAC1 (0.49) HDAC1HDAC3HDAC2NCOR2HDAC11
Succinic Acid SCHEMBL3948465 0.92 HDAC1 (0.57) HDAC1HDAC3HDAC2NCOR2HDAC11
Lactic Acid SCHEMBL3937225 0.91 HDAC1 (0.56) HDAC1HDAC3HDAC2NCOR2HDAC11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE40703-E1 Cell differentiation inducer, benzamide compounds SCHERING AKTIENGESELLSCHAFT (DE) 2009-04-28 US disclosed