SCHEMBL3940943

SCHEMBL3940943

CC(C)(C)Oc1cccc(CN2CCC(CCNC(=O)O)CC2)c1

nearest known ligand 0.58

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CHRM4 P08173 9/20 0.57
CHRM2 P08172 2/20 0.56
CHRM1 P11229 1/20 0.56
ACHE P22303 2/20 0.55
BCHE P06276 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3942812 0.90 CHRM4 (0.55) CHRM4ACHEBCHE
SCHEMBL3946316 0.89 CHRM4 (0.69) CHRM4CHRM2CHRM1
SCHEMBL2983017 0.85 CHRM4 (0.50) CHRM4CHRM2CHRM1ACHEBCHE
SCHEMBL3938451 0.82 CHRM4 (0.65) CHRM4ACHEBCHE
SCHEMBL3583996 0.80 CHRM4 (0.68) CHRM4CHRM2CHRM1
SCHEMBL5709492 0.79 CHRM4 (0.61) CHRM4CHRM2CHRM1
SCHEMBL3938442 0.79 CHRM4 (0.66) CHRM4CHRM2CHRM1ACHE
SCHEMBL3946379 0.79 MCHR1 (0.63) ACHE
SCHEMBL2980349 0.77 CHRM4 (0.51) CHRM4CHRM2ACHEBCHE
SCHEMBL5709518 0.77 OPRM1 (0.52) CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1720550-B1 DERIVATIVES OF PIPERIDINYLALKYLCARBAMATES, PREPARATION METHOD THEREOF AND USE OF SAME AS FAAH ENZYME INHIBITORS SANOFI AVENTIS (FR) 2009-04-15 EP claimed
EP-1720550-B1 DERIVATIVES OF PIPERIDINYLALKYLCARBAMATES, PREPARATION METHOD THEREOF AND USE OF SAME AS FAAH ENZYME INHIBITORS SANOFI AVENTIS (FR) 2009-04-15 EP disclosed
EP-1720550-A1 DERIVATIVES OF PIPERIDINYLALKYLCARBAMATES, PREPARATION METHOD THEREOF AND USE OF SAME AS FAAH ENZYME INHIBITORS Sanofi-Aventis (FR) 2006-11-15 EP disclosed
WO-2005089759-A1 DERIVATIVES OF PIPERIDINYLALKYLCARBAMATES, PREPARATION METHOD THEREOF AND USE OF SAME AS FAAH ENZYME INHIBITORS SANOFI-AVENTIS (FR) 2005-09-29 WO disclosed