SCHEMBL3942465

SCHEMBL3942465

CN(CC(O)c1ccc(O)cc1)C(=O)Oc1cnc(N(C)Cc2ccccc2)nc1-c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CASR P41180 4/20 0.41
PDK1 Q15118 5/20 0.37
CNR1 P21554 1/20 0.37
KDM4E B2RXH2 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
RPS6KB1 P23443 1/20 0.34
ACACB O00763 2/20 0.34
MTOR P42345 1/20 0.33
EGFR P00533 1/20 0.33
CSF1R P07333 1/20 0.33
PDK2 Q15119 1/20 0.33
PDK3 Q15120 1/20 0.33
PDK4 Q16654 1/20 0.33
ITGB1 P05556 1/20 0.33
ITGA4 P13612 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3946983 0.94 CASR (0.43) CASRPDK1CNR1KDM4EMEN1
SCHEMBL3945390 0.92 CASR (0.42) CASRCNR1KDM4EMEN1KMT2A
SCHEMBL4036518 0.92 CASR (0.40) CASRPDK1CNR1KDM4EMEN1
SCHEMBL3952113 0.91 CASR (0.44) CASRCNR1ACACB
SCHEMBL3947316 0.91 CASR (0.41) CASRPDK1CNR1MEN1KMT2A
SCHEMBL3945754 0.90 CASR (0.41) CASRCNR1KDM4EMEN1KMT2A
SCHEMBL3942446 0.87 CASR (0.41) CASRPDK1CNR1RPS6KB1ACACB
SCHEMBL3951654 0.86 CASR (0.41) CASRCNR1MEN1KMT2A
SCHEMBL3951537 0.85 CASR (0.46) CASRMEN1KMT2ACSF1R
SCHEMBL3945231 0.85 HPGD (0.40) CASRKDM4EMEN1KMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1718632-B1 PYRIMIDINE DERIVATIVES AS OREXIN RECEPTOR ANTAGONISTS SANOFI AVENTIS (FR) 2009-04-22 EP claimed