SCHEMBL3945231

SCHEMBL3945231

CN(CC(O)c1ccc2c(c1)OCO2)C(=O)Oc1cnc(N(C)Cc2ccccc2)nc1-c1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HPGD P15428 4/20 0.40
EDNRA P25101 3/20 0.39
CASR P41180 3/20 0.38
ALDH1A1 P00352 3/20 0.38
KDM4E B2RXH2 2/20 0.38
LMNA P02545 2/20 0.38
NPSR1 Q6W5P4 2/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
PTGFR P43088 2/20 0.37
TSHR P16473 2/20 0.36
GAA P10253 1/20 0.36
MAPT P10636 2/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
OGA O60502 1/20 0.36
HTT P42858 1/20 0.36
UBE2M P61081 1/20 0.35
DCUN1D1 Q96GG9 1/20 0.35
ADORA1 P30542 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3946983 0.87 CASR (0.43) CASRALDH1A1KDM4ESMN1; SMN2TSHR
SCHEMBL3942465 0.85 CASR (0.41) CASRKDM4ESMN1; SMN2MEN1KMT2A
SCHEMBL3947316 0.85 CASR (0.41) CASRLMNAMEN1KMT2A
SCHEMBL3942446 0.85 CASR (0.41) CASRLMNA
SCHEMBL3945390 0.84 CASR (0.42) CASRALDH1A1KDM4ELMNASMN1; SMN2
SCHEMBL4036518 0.84 CASR (0.40) CASRALDH1A1KDM4ENPSR1SMN1; SMN2
SCHEMBL3951654 0.84 CASR (0.41) CASRMAPTMEN1KMT2A
SCHEMBL3952113 0.84 CASR (0.44) CASRALDH1A1
SCHEMBL3951537 0.83 CASR (0.46) HPGDCASRALDH1A1MEN1KMT2A
SCHEMBL3945754 0.82 CASR (0.41) HPGDCASRALDH1A1KDM4ESMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1718632-B1 PYRIMIDINE DERIVATIVES AS OREXIN RECEPTOR ANTAGONISTS SANOFI AVENTIS (FR) 2009-04-22 EP claimed