SCHEMBL3945754

SCHEMBL3945754

CN(CC(O)c1ccc(C#N)cc1)C(=O)Oc1cnc(N(C)Cc2ccccc2)nc1-c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASR P41180 4/20 0.41
F2R P25116 1/20 0.40
NTRK1 P04629 1/20 0.38
NTRK3 Q16288 1/20 0.38
NTRK2 Q16620 1/20 0.38
ACACB O00763 1/20 0.37
SIGMAR1 Q99720 2/20 0.35
TMEM97 Q5BJF2 1/20 0.35
CNR1 P21554 1/20 0.35
KDM4E B2RXH2 2/20 0.35
ALDH1A1 P00352 1/20 0.35
HPGD P15428 1/20 0.35
CRHBP P24387 1/20 0.35
CRHR2 Q13324 1/20 0.35
CSNK2A1 P68400 1/20 0.34
EP300 Q09472 2/20 0.34
CTSA P10619 1/20 0.33
PTGDR2 Q9Y5Y4 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3946983 0.91 CASR (0.43) CASRACACBCNR1KDM4EALDH1A1
SCHEMBL3942465 0.90 CASR (0.41) CASRACACBCNR1KDM4EMEN1
SCHEMBL3945390 0.89 CASR (0.42) CASRCNR1KDM4EALDH1A1MEN1
SCHEMBL4036518 0.89 CASR (0.40) CASRCNR1KDM4EALDH1A1PTGDR2
SCHEMBL3952113 0.88 CASR (0.44) CASRACACBCNR1ALDH1A1
SCHEMBL3942446 0.84 CASR (0.41) CASRACACBCNR1RPS6KB1
SCHEMBL3947316 0.84 CASR (0.41) CASRCNR1MEN1KMT2ARPS6KB1
SCHEMBL3951654 0.83 CASR (0.41) CASRCNR1PTGDR2MEN1KMT2A
SCHEMBL3951537 0.83 CASR (0.46) CASRALDH1A1HPGDMEN1KMT2A
SCHEMBL3945231 0.82 HPGD (0.40) CASRKDM4EALDH1A1HPGDMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1718632-B1 PYRIMIDINE DERIVATIVES AS OREXIN RECEPTOR ANTAGONISTS SANOFI AVENTIS (FR) 2009-04-22 EP claimed