SCHEMBL394319

SCHEMBL394319

COC(=O)c1cnccc1N1CCSCC1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.47
ALDH1A1 P00352 4/20 0.47
GLA P06280 2/20 0.47
GAA P10253 2/20 0.47
F10 P00742 2/20 0.43
MAPT P10636 4/20 0.43
LMNA P02545 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
HSD17B10 Q99714 3/20 0.38
HTT P42858 2/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
HPGD P15428 1/20 0.37
CASP1 P29466 1/20 0.37
CASP7 P55210 1/20 0.37
NCOA1 Q15788 1/20 0.37
RCE1 Q9Y256 1/20 0.37
NCOA3 Q9Y6Q9 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20604844 0.83 PIM1 (0.48) KDM4EALDH1A1GLAGAAF10
SCHEMBL398926 0.82 KDM4C (0.41) KDM4EALDH1A1F10MAPTL3MBTL1
SCHEMBL2122533 0.80 CHIA (0.43) MAPTLMNA
SCHEMBL32678014 0.79 F10 (0.49) KDM4EALDH1A1GLAGAAF10
SCHEMBL32678012 0.79 F10 (0.49) KDM4EALDH1A1GLAGAAF10
SCHEMBL32678004 0.79 F10 (0.54) KDM4EALDH1A1GLAGAAF10
SCHEMBL28697754 0.74 MAPT (0.43) KDM4EALDH1A1GLAGAAF10
SCHEMBL9911009 0.74 KDM4E (0.51) KDM4EALDH1A1GLAGAAMAPT
SCHEMBL15714571 0.74 MYC (0.62) KDM4EALDH1A1GLAGAALMNA
SCHEMBL19943248 0.72 MAPT (0.55) KDM4EALDH1A1GAAMAPTL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2408745-A1 PIPERIDINE DERIVATIVES AS NK3 RECEPTOR ANTAGONISTS F. Hoffmann-La Roche AG (CH) 2012-01-25 EP disclosed