SCHEMBL3944151

SCHEMBL3944151

Cc1ccc(NC(=O)c2cccc(NC(=O)N(C)C)c2)cc1C(=O)Nc1cccnc1

nearest known ligand 0.77

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
BRAF P15056 14/20 0.77
CSF1R P07333 7/20 0.70
KIT P10721 1/20 0.62
KDR P35968 1/20 0.62
MAPK14 Q16539 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3934184 0.87 BRAF (1.00) BRAFCSF1RKITKDRMAPK14
SCHEMBL3937779 0.87 BRAF (1.00) BRAFCSF1RKITKDRMAPK14
SCHEMBL1276903 0.85 BRAF (1.00) BRAFCSF1R
SCHEMBL3942520 0.85 BRAF (1.00) BRAFCSF1RKITKDRMAPK14
SCHEMBL3943358 0.85 BRAF (0.80) BRAFCSF1RKITKDRMAPK14
SCHEMBL3945794 0.85 BRAF (0.80) BRAFCSF1RKITKDRMAPK14
SCHEMBL3937724 0.84 CSF1R (0.83) BRAFCSF1RKITKDRMAPK14
SCHEMBL3934972 0.84 BRAF (0.78) BRAFCSF1RKITKDRMAPK14
SCHEMBL27720443 0.83 BRAF (0.74) BRAFCSF1RKITKDRMAPK14
SCHEMBL3933229 0.83 BRAF (0.80) BRAFCSF1RKITKDRMAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1831198-B1 PYRIDINE CARBOXAMIDE DERIVATIVES FOR USE AS ANTICANCER AGENTS ASTRAZENECA AB (SE) 2009-04-08 EP disclosed
CN-101128454-A Pyridine carboxamide derivatives for use as anticancer agents ASTRAZENECA AB (SE) 2008-02-20 CN disclosed