SCHEMBL3937779

SCHEMBL3937779

Cc1cccc(C(=O)Nc2ccc(C)c(C(=O)Nc3cccnc3)c2)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
BRAF P15056 14/20 1.00
CSF1R P07333 6/20 0.80
KIT P10721 1/20 0.67
KDR P35968 1/20 0.67
MAPK14 Q16539 1/20 0.67
KCNK3 O14649 1/20 0.62
KCNK9 Q9NPC2 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3941714 0.91 BRAF (0.83) BRAFCSF1RKITKDRMAPK14
SCHEMBL3943800 0.89 BRAF (0.80) BRAFCSF1R
SCHEMBL12979 0.89 BRAF (0.79) BRAFCSF1RKCNK3KCNK9
SCHEMBL31661935 0.89 BRAF (0.79) BRAFCSF1RKCNK3KCNK9
SCHEMBL3935559 0.89 BRAF (0.80) BRAFCSF1RKCNK3KCNK9
SCHEMBL3941840 0.89 CSF1R (1.00) BRAFCSF1RKCNK3KCNK9
SCHEMBL3945794 0.89 BRAF (0.80) BRAFCSF1RKITKDRMAPK14
SCHEMBL3942520 0.89 BRAF (1.00) BRAFCSF1RKITKDRMAPK14
SCHEMBL1276903 0.89 BRAF (1.00) BRAFCSF1R
SCHEMBL3943358 0.89 BRAF (0.80) BRAFCSF1RKITKDRMAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1831198-B1 PYRIDINE CARBOXAMIDE DERIVATIVES FOR USE AS ANTICANCER AGENTS ASTRAZENECA AB (SE) 2009-04-08 EP disclosed
CN-101128454-A Pyridine carboxamide derivatives for use as anticancer agents ASTRAZENECA AB (SE) 2008-02-20 CN disclosed