SCHEMBL3945184

SCHEMBL3945184

COc1cccc(OCCC2CCCCN2)c1-c1cc(Cl)nc(N)n1

nearest known ligand 0.60

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 5/20 0.60
HSP90AB1 P08238 4/20 0.60
PIM1 P11309 1/20 0.42
PIM2 Q9P1W9 1/20 0.42
SSTR2 P30874 4/20 0.40
CHRNB4 P30926 1/20 0.40
CHRNA3 P32297 1/20 0.40
ADCY10 Q96PN6 1/20 0.39
CHRNA7 P36544 1/20 0.39
CYP1A2 P05177 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C19 P33261 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
HIF1A Q16665 1/20 0.38
PHLPP2 Q6ZVD8 1/20 0.38
NPY1R P25929 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4221151 0.78 HSP90AA1 (0.65) HSP90AA1HSP90AB1ADCY10
SCHEMBL3951313 0.77 HSP90AA1 (1.00) HSP90AA1HSP90AB1ADCY10CHRNA7
SCHEMBL7794951 0.76 CHRNB4 (0.47) PIM1PIM2SSTR2CHRNB4CHRNA3
SCHEMBL11449105 0.75 CHRNB4 (0.68) PIM1PIM2CHRNB4CHRNA3
SCHEMBL3951667 0.74 ADCY10 (0.63) HSP90AA1HSP90AB1ADCY10CYP2D6
SCHEMBL3946201 0.74 HSP90AA1 (0.65) HSP90AA1HSP90AB1ADCY10CHRNA7
SCHEMBL3944544 0.74 HSP90AA1 (0.76) HSP90AA1HSP90AB1ADCY10CHRNA7
SCHEMBL7794880 0.74 CHRNB4 (0.44) HSP90AA1HSP90AB1PIM1PIM2SSTR2
SCHEMBL7796351 0.73 CHRNB4 (0.40) HSP90AA1HSP90AB1PIM1PIM2SSTR2
SCHEMBL7792222 0.73 CHRNB4 (0.51) PIM1PIM2CHRNB4CHRNA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2049497-A2 PYRIMIDINE DERIVATIVES AS HSP90 INHIBITORS Astex Therapeutics Limited (GB) 2009-04-22 EP disclosed
WO-2006123165-A2 PYRIMIDINE DERIVATIVES AS HSP90 INHIBITORS ASTEX THERAPEUTICS LIMITED (GB) 2006-11-23 WO disclosed