SCHEMBL3945890

SCHEMBL3945890

CC(=O)N(NCc1cccc(F)c1Cl)C(COC(=O)Nc1cc2cc(F)ccc2cn1)CC(=O)NC[C@@H](N)CO.CC(=O)N(NCc1cccc(F)c1Cl)[C@H](COC(=O)Nc1cc2cc(F)ccc2cn1)CC(=O)NC[C@H](CO)NC(=O)OC(C)(C)C

nearest known ligand 0.31

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CDK9 P50750 1/20 0.31
SCN9A Q15858 2/20 0.30
CYP3A4 P08684 1/20 0.30
SCN10A Q9Y5Y9 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2877969 1.00 CDK9 (0.31) CDK9SCN9ACYP3A4SCN10A
SCHEMBL211003 0.97 CDK9 (0.32) CDK9SCN9ACYP3A4SCN10A
SCHEMBL213724 0.93 ABL1 (0.32)
SCHEMBL212277 0.91 CDK9 (0.32) CDK9SCN9ACYP3A4SCN10A
SCHEMBL210996 0.87 GSK3B (0.33) CDK9SCN9ACYP3A4SCN10A
SCHEMBL211004 0.87 SCN9A (0.33) CDK9SCN9ACYP3A4SCN10A
SCHEMBL212989 0.87 ABL1 (0.31)
SCHEMBL211097 0.86 MET (0.36) CDK9
SCHEMBL15808666 0.86
SCHEMBL211802 0.86 SYK (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009023193-A1 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS CYTOKINETICS, INCORPORATED (US) 2009-02-19 WO disclosed