SCHEMBL3947555

SCHEMBL3947555

O=C(O)C[C@H]1CCc2cc(OS(=O)(=O)C(F)(F)F)ccc21

nearest known ligand 0.65

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PPARD Q03181 19/20 0.65
PPARA Q07869 8/20 0.65
FFAR1 O14842 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9979558 0.86 PPARD (0.53) PPARDPPARAFFAR1
SCHEMBL14137078 0.84 ITGB3 (0.56) PPARDPPARA
SCHEMBL820621 0.81 PPARD (0.80) PPARDPPARA
SCHEMBL2995086 0.81 PPARD (0.80) PPARDPPARA
SCHEMBL20235187 0.81 PPARD (0.67) PPARDPPARAFFAR1
SCHEMBL821101 0.81 PPARD (0.80) PPARDPPARA
SCHEMBL3954189 0.81 PPARD (0.49) PPARDPPARAFFAR1
SCHEMBL4760401 0.79 PPARD (0.46) PPARDPPARAFFAR1
SCHEMBL6220392 0.79 PPARD (0.88) PPARDPPARAFFAR1
SCHEMBL12214666 0.79 PPARD (0.75) PPARDPPARAFFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1697333-A4 (3,4-DISUBSTITUTED)PROPANOIC CARBOXYLATES AS S1P (EDG) RECEPTOR AGONISTS MERCK & CO INC (US) 2009-07-08 EP disclosed
EP-1697333-A1 (3,4-DISUBSTITUTED)PROPANOIC CARBOXYLATES AS S1P (EDG) RECEPTOR AGONISTS Merck & Co., Inc. (US) 2006-09-06 EP disclosed
WO-2005058848-A1 (3,4-DISUBSTITUTED)PROPANOIC CARBOXYLATES AS S1P (EDG) RECEPTOR AGONISTS MERCK & CO., INC. (US) 2005-06-30 WO disclosed