SCHEMBL3947871

SCHEMBL3947871

COC(CNC(=O)OC(C)(C)C)c1ncc(F)cc1F

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR3 Q99500 1/20 0.39
SERPINE1 P05121 1/20 0.38
AAK1 Q2M2I8 4/20 0.36
GFER P55789 1/20 0.36
HSD17B10 Q99714 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
IRAK4 Q9NWZ3 3/20 0.35
SCN9A Q15858 1/20 0.34
ITK Q08881 2/20 0.34
ALOX5AP P20292 1/20 0.34
FEN1 P39748 1/20 0.34
EGFR P00533 1/20 0.34
SYK P43405 1/20 0.34
STK17B O94768 1/20 0.34
STK17A Q9UEE5 1/20 0.34
CTSS P25774 1/20 0.34
CTSK P43235 1/20 0.34
PTPN1 P18031 1/20 0.34
MKNK2 Q9HBH9 1/20 0.34
PCSK9 Q8NBP7 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3939421 0.85 SERPINE1 (0.40) S1PR3SERPINE1AAK1GFERHSD17B10
SCHEMBL3944958 0.84 AGBL2 (0.38) S1PR3IRAK4
SCHEMBL24468300 0.76 S1PR3 (0.44) S1PR3AAK1HSD17B10SYKCTSS
SCHEMBL29685920 0.76 S1PR3 (0.44) S1PR3AAK1HSD17B10SYKCTSS
SCHEMBL31448001 0.73 AGBL2 (0.32)
SCHEMBL3938021 0.73 AGBL2 (0.32)
SCHEMBL31569062 0.72 AAK1 (0.35) SERPINE1AAK1GFERHSD17B10L3MBTL1
SCHEMBL1395922 0.70 TAAR1 (0.33)
SCHEMBL5456915 0.70 SYK (0.46) S1PR3AAK1IRAK4SYK
SCHEMBL30411121 0.70 MKNK2 (0.42) SERPINE1AAK1SYKMKNK2PCSK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009095712-A2 CHEMICAL COMPOUNDS ASTRAZENECA AB (SE) 2009-08-06 WO disclosed
WO-2009016410-A2 CHEMICAL COMPOUNDS 831 ASTRAZENECA AB (SE) 2009-02-05 WO disclosed
WO-2008132502-A1 PYRAZOLYL-AMINO-SUBSTITUTED PYRIMIDINES AND THEIR USE FOR THE TREATMENT OF CANCER ASTRAZENECA AB (SE) 2008-11-06 WO disclosed