SCHEMBL3948611

SCHEMBL3948611

Cc1ccc(S(=O)(=O)OC[C@@H]2CNC(=O)O2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.53
MAOA P21397 1/20 0.53
SLC6A2 P23975 1/20 0.53
PKM P14618 1/20 0.52
MAPT P10636 2/20 0.44
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
ALDH1A1 P00352 4/20 0.43
CYP3A4 P08684 3/20 0.43
CYP2D6 P10635 2/20 0.43
TSHR P16473 2/20 0.43
MAPK1 P28482 2/20 0.43
CYP2C9 P11712 2/20 0.43
CYP2C19 P33261 2/20 0.43
USP2 O75604 1/20 0.40
HPGD P15428 1/20 0.40
HSD17B10 Q99714 1/20 0.40
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37
CA9 Q16790 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7540998 1.00 LMNA (0.53) LMNAMAOASLC6A2PKMMAPT
SCHEMBL3950063 1.00 LMNA (0.53) LMNAMAOASLC6A2PKMMAPT
SCHEMBL5309585 0.84 LMNA (0.52) LMNAMAOASLC6A2PKMMAPT
SCHEMBL14167936 0.83 PRMT5 (0.49) LMNAMAOASLC6A2PKMMAPT
SCHEMBL4777682 0.81 ALDH1A1 (0.39) LMNAMAOASLC6A2PKMMAPT
SCHEMBL14290873 0.81 ALDH1A1 (0.39) LMNAMAOASLC6A2PKMMAPT
SCHEMBL439063 0.77 PRMT5 (0.54) LMNAPKMMAPTMEN1KMT2A
SCHEMBL439062 0.77 PRMT5 (0.54) LMNAPKMMAPTMEN1KMT2A
SCHEMBL450879 0.77 PRMT5 (0.54) LMNAPKMMAPTMEN1KMT2A
SCHEMBL22107643 0.77 LMNA (0.51) LMNAMAOASLC6A2PKMMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1833977-B1 ENANTIOCONVERGENT CHEMOENZYMATIC SYNTHESIS OF (R)- GAMMA-AMINO-BETA-HYDROXYBUTYRIC ACID ((R) - GABOB) COUNCIL SCIENT IND RES (IN) 2009-04-29 EP claimed
US-7374926-B2 Enantioconvergent chemoenzymatic synthesis of (R)-γ-amino-β-hydroxybutyric acid ((R)-GABOB) COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH (IN) 2008-05-20 US claimed
EP-1833977-A1 ENANTIOCONVERGENT CHEMOENZYMATIC SYNTHESIS OF (R)- GAMMA-AMINO-BETA-HYDROXYBUTYRIC ACID ((R) -GABOB) COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2007-09-19 EP claimed
US-20060141606-A1 Enantioconvergent chemoenzymatic synthesis of (R)-gamma-amino-beta-hydroxybutyric acid ((R)-GABOB) COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH (IN) 2006-06-29 US claimed
WO-2006064513-A1 ENANTIOCONVERGENT CHEMOENZYMATIC SYNTHESIS OF (R)- GAMMA-AMINO-BETA-HYDROXYBUTYRIC ACID ((R) -GABOB) COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2006-06-22 WO claimed
JP-62108870-A None JP disclosed
WO-2025026997-A1 SUBSTITUED BICYCLIC HETEROCYCLIC YAP-TEAD AND/OR TAZ-TEAD INHIBITORS MERCK PATENT GMBH (DE) 2025-02-06 WO disclosed
EP-1833977-B1 ENANTIOCONVERGENT CHEMOENZYMATIC SYNTHESIS OF (R)- GAMMA-AMINO-BETA-HYDROXYBUTYRIC ACID ((R) - GABOB) COUNCIL SCIENT IND RES (IN) 2009-04-29 EP disclosed
EP-1833977-B1 ENANTIOCONVERGENT CHEMOENZYMATIC SYNTHESIS OF (R)- GAMMA-AMINO-BETA-HYDROXYBUTYRIC ACID ((R) - GABOB) COUNCIL SCIENT IND RES (IN) 2009-04-29 EP disclosed
US-7374926-B2 Enantioconvergent chemoenzymatic synthesis of (R)-γ-amino-β-hydroxybutyric acid ((R)-GABOB) COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH (IN) 2008-05-20 US disclosed
US-7374926-B2 Enantioconvergent chemoenzymatic synthesis of (R)-γ-amino-β-hydroxybutyric acid ((R)-GABOB) COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH (IN) 2008-05-20 US disclosed
US-7374926-B2 Enantioconvergent chemoenzymatic synthesis of (R)-γ-amino-β-hydroxybutyric acid ((R)-GABOB) COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH (IN) 2008-05-20 US disclosed
EP-1833977-A1 ENANTIOCONVERGENT CHEMOENZYMATIC SYNTHESIS OF (R)- GAMMA-AMINO-BETA-HYDROXYBUTYRIC ACID ((R) -GABOB) COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2007-09-19 EP disclosed
US-20060141606-A1 Enantioconvergent chemoenzymatic synthesis of (R)-gamma-amino-beta-hydroxybutyric acid ((R)-GABOB) COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH (IN) 2006-06-29 US disclosed
WO-2006064513-A1 ENANTIOCONVERGENT CHEMOENZYMATIC SYNTHESIS OF (R)- GAMMA-AMINO-BETA-HYDROXYBUTYRIC ACID ((R) -GABOB) COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2006-06-22 WO disclosed
JP-S62108870-A OPTICALLY ACTIVE 5-SULFONYLOXYMETHYL-2-OXAZOLIDINONE DERIVATIVE AND PRODUCTION THEREOF KANEGAFUCHI CHEM IND CO LTD 1987-05-20 JP disclosed