SCHEMBL3948975

SCHEMBL3948975

NCCc1ccc(C2CCC2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 2/20 0.49
NUDT1 P36639 1/20 0.49
TAAR1 Q96RJ0 7/20 0.45
HTR2A P28223 3/20 0.45
CYP2A6 P11509 2/20 0.45
CYP1A2 P05177 1/20 0.45
KDM4E B2RXH2 1/20 0.45
ALDH1A1 P00352 1/20 0.45
HTR1A P08908 1/20 0.45
ADRA2A P08913 1/20 0.45
SLC6A2 P23975 1/20 0.45
CYP2C19 P33261 1/20 0.45
HTR3A P46098 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
SPHK1 Q9NYA1 1/20 0.45
HTR1D P28221 2/20 0.44
BLM P54132 1/20 0.43
KMT2A Q03164 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4363948 0.94 BACE1 (0.56) BACE1NUDT1TAAR1HTR2ACYP2A6
SCHEMBL14452295 0.91 SPHK1 (0.51) BACE1NUDT1TAAR1HTR2ACYP2A6
SCHEMBL11997346 0.83 HRH3 (0.44) SPHK1LOXL2
SCHEMBL28258215 0.82 SLC18A3 (0.52) BACE1TAAR1HTR2ACYP2A6CYP1A2
SCHEMBL3946982 0.81 NUDT1 (0.38) BACE1NUDT1TAAR1CYP2A6CYP1A2
SCHEMBL7926837 0.80 GFER (0.54) BACE1NUDT1ALDH1A1SPHK1HTR1D
SCHEMBL28672856 0.80 HTR3A (0.56) HTR3A
SCHEMBL19212128 0.80 LSS (0.55) TAAR1CYP2A6CYP1A2CYP2C19SPHK1
SCHEMBL16671443 0.79 SPHK1 (0.57) HTR2ASPHK1
SCHEMBL10232991 0.78 HRH3 (0.44) BACE1NUDT1SPHK1HTR1DLOXL2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2051967-A1 BENZIMIDAZOLE DERIVATIVES USEFUL IN TREATMENT OF VALLINOID RECEPTOR TRPV1 RELATED DISORDERS AstraZeneca AB (SE) 2009-04-29 EP disclosed
WO-2008018827-A1 BENZIMIDAZOLE DERIVATIVES USEFUL IN TREATMENT OF VALLINOID RECEPTOR TRPV1 RELATED DISORDERS ASTRAZENECA AB (SE) 2008-02-14 WO disclosed