SCHEMBL3949028

SCHEMBL3949028

Clc1ccc(CNc2cnccn2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 1.00
KDM4E B2RXH2 6/20 1.00
HPGD P15428 5/20 0.71
KMT2A Q03164 2/20 0.70
MEN1 O00255 1/20 0.70
CYP1A2 P05177 2/20 0.65
CYP2C9 P11712 2/20 0.65
CYP2C19 P33261 2/20 0.65
CYP2D6 P10635 1/20 0.65
POLB P06746 1/20 0.58
DYRK1A Q13627 1/20 0.55
CLK4 Q9HAZ1 1/20 0.55
NPSR1 Q6W5P4 1/20 0.54
HDAC1 Q13547 2/20 0.50
HDAC6 Q9UBN7 2/20 0.50
HDAC8 Q9BY41 1/20 0.50
NPC1 O15118 1/20 0.49
GAA P10253 1/20 0.49
MAPT P10636 1/20 0.49
RAB9A P51151 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3952458 0.84 ALDH1A1 (0.77) ALDH1A1KDM4EHPGDKMT2AMEN1
SCHEMBL18448724 0.83 KDM4E (0.71) ALDH1A1KDM4EHPGDKMT2AMEN1
SCHEMBL30352430 0.83 KDM4E (0.71) ALDH1A1KDM4EHPGDKMT2AMEN1
SCHEMBL4141061 0.83 ALDH1A1 (1.00) ALDH1A1KDM4EHPGDKMT2AMEN1
SCHEMBL3956196 0.83 ALDH1A1 (1.00) ALDH1A1KDM4EHPGDKMT2AMEN1
SCHEMBL23780412 0.83 ALDH1A1 (0.71) ALDH1A1KDM4EHPGDKMT2AMEN1
SCHEMBL14075916 0.83 ALDH1A1 (0.71) ALDH1A1KDM4EHPGDKMT2AMEN1
SCHEMBL3953451 0.82 ALDH1A1 (1.00) ALDH1A1KDM4EHPGDKMT2AMEN1
SCHEMBL3956255 0.81 ALDH1A1 (0.68) ALDH1A1KDM4EHPGDKMT2AMEN1
SCHEMBL29999485 0.79 ALDH1A1 (0.69) ALDH1A1KDM4EHPGDKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024155555-A1 NEUROPROTECTIVE COMPOUNDS FOR THERAPEUTIC USE NIMML INSTITUTE (US) 2024-07-25 WO disclosed
WO-2009029617-A1 DIARYLAMINE-SUBSTITUTED QUINOLONES USEFUL AS INDUCIBLE NITRIC OXIDE SYNTHASE INHIBITORS KALYPSYS, INC. (US) 2009-03-05 WO disclosed
EP-0124155-B1 PYRAZINE COMPOUNDS, THEIR PREPARATION AND THEIR USE, COMPOSITIONS CONTAINING THEM AND METHOD OF COMBATING UNDESIRED PLANT GROWTH SHELL INTERNATIONALE RESEARCHMAATSCHAPPIJ B.V. (NL) 1987-06-03 EP disclosed
EP-0124155-A1 Pyrazine compounds, their preparation and their use, compositions containing them and method of combating undesired plant growth SHELL INTERNATIONALE RESEARCHMAATSCHAPPIJ B.V. (NL) 1984-11-07 EP disclosed
US-4441912-A N-Pyrazinyl-N-benzylcarbamates, having fungicidal and plant growth regulating properties SHELL OIL COMPANY (US) 1984-04-10 US disclosed
US-4359576-A N-Pyrazinyl-N-benzylcarbamates, having fungicidal and plant growth regulating properties SHELL OIL COMPANY (US) 1982-11-16 US disclosed