SCHEMBL3953451

SCHEMBL3953451

c1ccc(CNc2cnccn2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 1.00
HPGD P15428 4/20 1.00
MEN1 O00255 1/20 1.00
KMT2A Q03164 1/20 1.00
KDM4E B2RXH2 6/20 0.70
FABP1 P07148 1/20 0.65
FABP6 P51161 1/20 0.65
CYP1A2 P05177 3/20 0.64
CYP2D6 P10635 3/20 0.64
CYP2C19 P33261 2/20 0.64
CYP2C9 P11712 1/20 0.64
CXCR4 P61073 1/20 0.56
NOS2 P35228 1/20 0.56
CYP3A4 P08684 2/20 0.54
CLK4 Q9HAZ1 2/20 0.54
USP2 O75604 1/20 0.54
HSD17B10 Q99714 1/20 0.52
LTA4H P09960 1/20 0.51
HDAC1 Q13547 1/20 0.49
HDAC8 Q9BY41 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3948160 0.87 ALDH1A1 (0.77) ALDH1A1HPGDMEN1KMT2AKDM4E
SCHEMBL3952458 0.87 ALDH1A1 (0.77) ALDH1A1HPGDMEN1KMT2AKDM4E
SCHEMBL5766313 0.85 ALDH1A1 (0.73) ALDH1A1HPGDMEN1KMT2AKDM4E
SCHEMBL3949028 0.82 ALDH1A1 (1.00) ALDH1A1HPGDMEN1KMT2AKDM4E
SCHEMBL14075916 0.82 ALDH1A1 (0.71) ALDH1A1HPGDMEN1KMT2AKDM4E
SCHEMBL23780412 0.82 ALDH1A1 (0.71) ALDH1A1HPGDMEN1KMT2AKDM4E
SCHEMBL4141061 0.82 ALDH1A1 (1.00) ALDH1A1HPGDMEN1KMT2AKDM4E
SCHEMBL3956196 0.82 ALDH1A1 (1.00) ALDH1A1HPGDMEN1KMT2AKDM4E
SCHEMBL3956283 0.82 ALDH1A1 (0.70) ALDH1A1HPGDMEN1KMT2AKDM4E
SCHEMBL3957528 0.80 ALDH1A1 (0.68) ALDH1A1HPGDMEN1KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3326715-B1 OXALIC ACID MONOAMIDE LIGAND, AND USES THEREOF IN COUPLING REACTION OF COPPER-CATALYZED ARYL HALOGEN SUBSTITUTE CE PHARM CO LTD (CN) 2021-09-15 EP disclosed
US-20180207628-A1 OXALIC ACID MONOAMIDE LIGAND, AND USES THEREOF IN COUPLING REACTION OF COPPER-CATALYZED ARYL HALOGEN SUBSTITUTE SHANGHAI INSTITUTE OF ORGANIC CHEMISTRY, CHINESE ACADEMY OF SCIENCES (CN) 2018-07-26 US disclosed
US-20180207628-A1 OXALIC ACID MONOAMIDE LIGAND, AND USES THEREOF IN COUPLING REACTION OF COPPER-CATALYZED ARYL HALOGEN SUBSTITUTE SHANGHAI INSTITUTE OF ORGANIC CHEMISTRY, CHINESE ACADEMY OF SCIENCES (CN) 2018-07-26 US disclosed
EP-3326715-A1 OXALIC ACID MONOAMIDE LIGAND, AND USES THEREOF IN COUPLING REACTION OF COPPER-CATALYZED ARYL HALOGEN SUBSTITUTE Shanghai Institute of Organic Chemistry, Chinese Academy of Sciences (CN) 2018-05-30 EP disclosed
WO-2009029617-A1 DIARYLAMINE-SUBSTITUTED QUINOLONES USEFUL AS INDUCIBLE NITRIC OXIDE SYNTHASE INHIBITORS KALYPSYS, INC. (US) 2009-03-05 WO disclosed
US-RE30563-E Preparation of benzoylureas ELI LILLY AND COMPANY (US) 1981-03-31 US disclosed
US-4133956-A Preparation of benzoylureas ELI LILLY AND COMPANY (US) 1979-01-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180207628-A1 OXALIC ACID MONOAMIDE LIGAND, AND USES THEREOF IN COUPLING REACTION OF COPPER-CATALYZED ARYL HALOGEN SUBSTITUTE AOC2, AOC1, AOC3 ALDH1A1 213/4885HPGD 1526/4885MEN1 388/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.