SCHEMBL3949634

SCHEMBL3949634

CC(NC(=O)c1ccccc1)C(C)C(=O)N1CCC(O)(c2ccc(Cl)cc2Cl)CC1

nearest known ligand 0.61

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 16/20 0.61
CYP3A4 P08684 2/20 0.46
UGCG Q16739 2/20 0.46
EPHX2 P34913 1/20 0.45
ACE2 Q9BYF1 1/20 0.44
KCNH2 Q12809 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12398377 0.88 CCR1 (0.74) CCR1KCNH2
SCHEMBL2160124 0.88 CCR1 (0.74) CCR1KCNH2
SCHEMBL3941668 0.86 CCR1 (0.78) CCR1ACE2KCNH2
SCHEMBL10291673 0.78 CCR1 (0.45) CCR1CYP3A4UGCGEPHX2
SCHEMBL3945220 0.78 CCR1 (0.78) CCR1ACE2
SCHEMBL3946317 0.78 CCR1 (0.78) CCR1ACE2
SCHEMBL3007113 0.76 CCR1 (1.00) CCR1
SCHEMBL3943809 0.76 CCR1 (1.00) CCR1
SCHEMBL3007118 0.76 CCR1 (1.00) CCR1
SCHEMBL3940996 0.76 CCR1 (0.67) CCR1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2049486-A2 PIPERIDINYL DERIVATIVES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY Bristol-Myers Squibb Company (US) 2009-04-22 EP disclosed
WO-2007092681-A2 PIPERIDINYL DERIVATIVES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY BRISTOL-MYERS SQUIBB COMPANY (US) 2007-08-16 WO disclosed